Search Results - "Atkinson SJ"

Using qualitative risk assessment to re-evaluate the veterinary fence paradigm within the Kavango Zambezi Transfrontier Conservation Area.

Authors: Rosen LE Atkinson SJ Babayani ND et al.

Source: Frontiers in veterinary science [Front Vet Sci] 2026 Jan 30; Vol. 12, pp. 1702631. Date of Electronic Publication: 2026 Jan 30 (Print Publication: 2025).

Publication Type: Journal Article

Journal Info: Publisher: Frontiers Media S.A Country of Publication: Switzerland NLM ID: 101666658 Publication Model: eCollection Cited Medium: Print ISSN: 2297-1769 (Print) Linking ISSN: 22971769 NLM ISO Abbreviation: Front Vet Sci Subsets: PubMed not MEDLINE

BET Isoform Selectivity through Diverse Linkers for Bivalent Inhibitors: GSK785, a BRD2/4-Selective Bivalent BET Inhibitor.

Authors: Rianjongdee F Atkinson SJ Bamborough P et al.

Source: Journal of medicinal chemistry [J Med Chem] 2026 Jan 22; Vol. 69 (2), pp. 895-917. Date of Electronic Publication: 2025 Dec 30.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Mechanistic safety assessment via multi-omic characterisation of systemic pathway perturbations following in vivo MAT2A inhibition.

Authors: Fogal V Michopoulos F Jarnuczak AF et al.

Source: Archives of toxicology [Arch Toxicol] 2024 Aug; Vol. 98 (8), pp. 2589-2603. Date of Electronic Publication: 2024 May 17.

Publication Type: Journal Article

Journal Info: Publisher: Springer-Verlag Country of Publication: Germany NLM ID: 0417615 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1432-0738 (Electronic) Linking ISSN: 03405761 NLM ISO Abbreviation: Arch Toxicol Subsets: MEDLINE

Phenotype-Led Identification of IL-10 Upregulators in Human CD4⁺ T-cells and Elucidation of Their Pharmacology as Highly Selective CDK8/CDK19 Inhibitors.

Authors: Nicolle S Barker M Barrett J et al.

Source: Journal of medicinal chemistry [J Med Chem] 2025 Jan 23; Vol. 68 (2), pp. 1883-1900. Date of Electronic Publication: 2025 Jan 08.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Sulfotransferase 1C2 Increases Mitochondrial Respiration by Converting Mitochondrial Membrane Cholesterol to Cholesterol Sulfate.

Authors: Kolb AJ Corridon P Ullah M et al.

Source: Biochemistry [Biochemistry] 2024 Sep 17; Vol. 63 (18), pp. 2310-2322. Date of Electronic Publication: 2024 Aug 28.

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 0370623 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4995 (Electronic) Linking ISSN: 00062960 NLM ISO Abbreviation: Biochemistry Subsets: MEDLINE

Development of a Series of Pyrrolopyridone MAT2A Inhibitors.

Authors: Atkinson SJ Bagal SK Argyrou A et al.

Source: Journal of medicinal chemistry [J Med Chem] 2024 Mar 28; Vol. 67 (6), pp. 4541-4559. Date of Electronic Publication: 2024 Mar 11.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Selective Phosphodiesterase 1 Inhibitor BTTQ Reduces Blood Pressure in Spontaneously Hypertensive and Dahl Salt Sensitive Rats: Role of Peripheral Vasodilation.

Authors: Dey AB Khedr S Bean J et al.

Source: Frontiers in physiology [Front Physiol] 2020 Sep 08; Vol. 11, pp. 543727. Date of Electronic Publication: 2020 Sep 08 (Print Publication: 2020).

Publication Type: Journal Article

Journal Info: Publisher: Frontiers Research Foundation Country of Publication: Switzerland NLM ID: 101549006 Publication Model: eCollection Cited Medium: Print ISSN: 1664-042X (Print) Linking ISSN: 1664042X NLM ISO Abbreviation: Front Physiol Subsets: PubMed not MEDLINE

Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation.

Authors: Gilan O Rioja I Knezevic K et al.

Source: Science (New York, N.Y.) [Science] 2020 Apr 24; Vol. 368 (6489), pp. 387-394. Date of Electronic Publication: 2020 Mar 19.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Association for the Advancement of Science Country of Publication: United States NLM ID: 0404511 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1095-9203 (Electronic) Linking ISSN: 00368075 NLM ISO Abbreviation: Science Subsets: MEDLINE

Hypoxic cancer-associated fibroblasts increase NCBP2-AS2/HIAR to promote endothelial sprouting through enhanced VEGF signaling.

Authors: Kugeratski FG Atkinson SJ Neilson LJ et al.

Source: Science signaling [Sci Signal] 2019 Feb 05; Vol. 12 (567). Date of Electronic Publication: 2019 Feb 05.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Association for the Advancement of Science Country of Publication: United States NLM ID: 101465400 Publication Model: Electronic Cited Medium: Internet ISSN: 1937-9145 (Electronic) Linking ISSN: 19450877 NLM ISO Abbreviation: Sci Signal Subsets: MEDLINE

Kidney surveillance in the spotlight: contrast-induced acute kidney injury illuminated.

Authors: Atkinson SJ

Source: The Journal of clinical investigation [J Clin Invest] 2018 Jul 02; Vol. 128 (7), pp. 2754-2756. Date of Electronic Publication: 2018 Jun 04.

Publication Type: Journal Article; Comment

Journal Info: Publisher: American Society for Clinical Investigation Country of Publication: United States NLM ID: 7802877 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1558-8238 (Electronic) Linking ISSN: 00219738 NLM ISO Abbreviation: J Clin Invest Subsets: MEDLINE

The β3-integrin endothelial adhesome regulates microtubule-dependent cell migration.

Authors: Atkinson SJ Gontarczyk AM Alghamdi AA et al.

Source: EMBO reports [EMBO Rep] 2018 Jul; Vol. 19 (7). Date of Electronic Publication: 2018 May 24.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 100963049 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1469-3178 (Electronic) Linking ISSN: 1469221X NLM ISO Abbreviation: EMBO Rep Subsets: MEDLINE

A patent review of MAT2a inhibitors (2018-2021).

Authors: Atkinson SJ Evans L Scott JS

Source: Expert opinion on therapeutic patents [Expert Opin Ther Pat] 2022 Oct; Vol. 32 (10), pp. 1043-1053. Date of Electronic Publication: 2022 Sep 01.

Publication Type: Review; Journal Article

Journal Info: Publisher: Informa Healthcare Country of Publication: England NLM ID: 9516419 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1744-7674 (Electronic) Linking ISSN: 13543776 NLM ISO Abbreviation: Expert Opin Ther Pat Subsets: MEDLINE

Design, Synthesis, and Characterization of I-BET567, a Pan-Bromodomain and Extra Terminal (BET) Bromodomain Oral Candidate.

Authors: Humphreys PG Atkinson SJ Bamborough P et al.

Source: Journal of medicinal chemistry [J Med Chem] 2022 Feb 10; Vol. 65 (3), pp. 2262-2287. Date of Electronic Publication: 2022 Jan 07.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors.

Authors: Seal JT Atkinson SJ Bamborough P et al.

Source: Journal of medicinal chemistry [J Med Chem] 2021 Aug 12; Vol. 64 (15), pp. 10772-10805. Date of Electronic Publication: 2021 Jul 13.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Discovery of a Highly Selective BET BD2 Inhibitor from a DNA-Encoded Library Technology Screening Hit.

Authors: Rianjongdee F Atkinson SJ Chung CW et al.

Source: Journal of medicinal chemistry [J Med Chem] 2021 Aug 12; Vol. 64 (15), pp. 10806-10833. Date of Electronic Publication: 2021 Jul 12.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Identification of a Series of N-Methylpyridine-2-carboxamides as Potent and Selective Inhibitors of the Second Bromodomain (BD2) of the Bromo and Extra Terminal Domain (BET) Proteins.

Authors: Harrison LA Atkinson SJ Bassil A et al.

Source: Journal of medicinal chemistry [J Med Chem] 2021 Aug 12; Vol. 64 (15), pp. 10742-10771. Date of Electronic Publication: 2021 Jul 07.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors.

Authors: Lucas SCC Atkinson SJ Chung CW et al.

Source: Journal of medicinal chemistry [J Med Chem] 2021 Aug 12; Vol. 64 (15), pp. 10711-10741. Date of Electronic Publication: 2021 Jul 14.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Role of matrix metalloproteinase-8 as a mediator of injury in intestinal ischemia and reperfusion.

Authors: Daly MC Atkinson SJ Varisco BM et al.

Source: FASEB journal : official publication of the Federation of American Societies for Experimental Biology [FASEB J] 2016 Oct; Vol. 30 (10), pp. 3453-3460. Date of Electronic Publication: 2016 Jul 19.

Publication Type: Journal Article; Research Support, N.I.H., Extramural

Journal Info: Publisher: Federation of American Societies for Experimental Biology Country of Publication: United States NLM ID: 8804484 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1530-6860 (Electronic) Linking ISSN: 08926638 NLM ISO Abbreviation: FASEB J Subsets: MEDLINE

Matrix Metalloproteinase-8 Augments Bacterial Clearance in a Juvenile Sepsis Model.

Authors: Atkinson SJ Varisco BM Sandquist M et al.

Source: Molecular medicine (Cambridge, Mass.) [Mol Med] 2016 Oct; Vol. 22, pp. 455-463. Date of Electronic Publication: 2016 Aug 08.

Publication Type: Journal Article

Journal Info: Publisher: BioMed Central Country of Publication: England NLM ID: 9501023 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1528-3658 (Electronic) Linking ISSN: 10761551 NLM ISO Abbreviation: Mol Med Subsets: PubMed not MEDLINE

A wandering path toward prevention for acute kidney injury.

Authors: Atkinson SJ

Source: The Journal of clinical investigation [J Clin Invest] 2016 May 02; Vol. 126 (5), pp. 1640-2. Date of Electronic Publication: 2016 Apr 18.

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Comment

Journal Info: Publisher: American Society for Clinical Investigation Country of Publication: United States NLM ID: 7802877 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1558-8238 (Electronic) Linking ISSN: 00219738 NLM ISO Abbreviation: J Clin Invest Subsets: MEDLINE