Search Results - "Epplin MP"

Corrigendum to "A subunit-selective negative allosteric modulator of GluN1/GluN3A glycine-activated receptor" [Molecular Pharmacology 108 (2026) 100104].

Authors: Jacobs L Nguyen TT McCallum A et al.

Source: Molecular pharmacology [Mol Pharmacol] 2026 Apr; Vol. 108 (4), pp. 100118. Date of Electronic Publication: 2026 Mar 30.

Publication Type: Published Erratum

Journal Info: Publisher: American Society for Pharmacology and Experimental Therapeutics Country of Publication: Netherlands NLM ID: 0035623 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-0111 (Electronic) Linking ISSN: 0026895X NLM ISO Abbreviation: Mol Pharmacol Subsets: MEDLINE; In Process

A subunit-selective negative allosteric modulator of GluN1/GluN3A glycine-activated receptor.

Authors: Jacobs L Nguyen TT McCallum A et al.

Source: Molecular pharmacology [Mol Pharmacol] 2026 Mar; Vol. 108 (3), pp. 100104. Date of Electronic Publication: 2026 Jan 29.

Publication Type: Journal Article

Journal Info: Publisher: American Society for Pharmacology and Experimental Therapeutics Country of Publication: Netherlands NLM ID: 0035623 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-0111 (Electronic) Linking ISSN: 0026895X NLM ISO Abbreviation: Mol Pharmacol Subsets: MEDLINE

Discrete interneuron subsets participate in GluN1/GluN3A excitatory glycine receptor (eGlyR)-mediated regulation of hippocampal network activity throughout development and evolution.

Authors: Kim JH Vlachos A Mahadevan V et al.

Source: Research square [Res Sq] 2025 Oct 15. Date of Electronic Publication: 2025 Oct 15.

Publication Type: Journal Article; Preprint

Journal Info: Country of Publication: United States NLM ID: 101768035 Publication Model: Electronic Cited Medium: Internet ISSN: 2693-5015 (Electronic) Linking ISSN: 26935015 NLM ISO Abbreviation: Res Sq Subsets: PubMed not MEDLINE

Discrete interneuron subsets participate in GluN1/GluN3A excitatory glycine receptor (eGlyR)-mediated regulation of hippocampal network activity throughout development and evolution.

Authors: Kim JH Vlachos A Mahadevan V et al.

Source: BioRxiv : the preprint server for biology [bioRxiv] 2025 Sep 25. Date of Electronic Publication: 2025 Sep 25.

Publication Type: Journal Article; Preprint

Journal Info: Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE

Selective enhancement of the interneuron network and gamma-band power via GluN2C/GluN2D NMDA receptor potentiation.

Authors: Camp CR Banke TG Xing H et al.

Source: The Journal of physiology [J Physiol] 2025 Jul; Vol. 603 (14), pp. 4027-4049. Date of Electronic Publication: 2025 Jun 25.

Publication Type: Journal Article; Research Support, N.I.H., Extramural

Journal Info: Publisher: Cambridge Univ. Press Country of Publication: England NLM ID: 0266262 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1469-7793 (Electronic) Linking ISSN: 00223751 NLM ISO Abbreviation: J Physiol Subsets: MEDLINE

Selective Enhancement of the Interneuron Network and Gamma-Band Power via GluN2C/GluN2D NMDA Receptor Potentiation.

Authors: Camp CR Banke TG Xing H et al.

Source: BioRxiv : the preprint server for biology [bioRxiv] 2024 Nov 05. Date of Electronic Publication: 2024 Nov 05.

Publication Type: Journal Article; Preprint

Journal Info: Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE

Distinct GluN1 and GluN2 Structural Determinants for Subunit-Selective Positive Allosteric Modulation of N-Methyl-d-aspartate Receptors.

Authors: Strong KL Epplin MP Ogden KK et al.

Source: ACS chemical neuroscience [ACS Chem Neurosci] 2021 Jan 06; Vol. 12 (1), pp. 79-98. Date of Electronic Publication: 2020 Dec 16.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101525337 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1948-7193 (Electronic) Linking ISSN: 19487193 NLM ISO Abbreviation: ACS Chem Neurosci Subsets: MEDLINE

Negative allosteric modulation of GluN1/GluN3 NMDA receptors.

Authors: Zhu Z Yi F Epplin MP et al.

Source: Neuropharmacology [Neuropharmacology] 2020 Oct 01; Vol. 176, pp. 108117. Date of Electronic Publication: 2020 May 07.

Publication Type: Journal Article; Research Support, N.I.H., Extramural

Journal Info: Publisher: Pergamon Press Country of Publication: England NLM ID: 0236217 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-7064 (Electronic) Linking ISSN: 00283908 NLM ISO Abbreviation: Neuropharmacology Subsets: MEDLINE

Discovery of Dihydropyrrolo[1,2-a]pyrazin-3(4H)-one-Based Second-Generation GluN2C- and GluN2D-Selective Positive Allosteric Modulators (PAMs) of the N-Methyl-d-Aspartate (NMDA) Receptor.

Authors: Epplin MP Mohan A Harris LD et al.

Source: Journal of medicinal chemistry [J Med Chem] 2020 Jul 23; Vol. 63 (14), pp. 7569-7600. Date of Electronic Publication: 2020 Jul 06.

Publication Type: Journal Article; Research Support, N.I.H., Extramural

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Biased modulators of NMDA receptors control channel opening and ion selectivity.

Authors: Perszyk RE Swanger SA Shelley C et al.

Source: Nature chemical biology [Nat Chem Biol] 2020 Feb; Vol. 16 (2), pp. 188-196. Date of Electronic Publication: 2020 Jan 20.

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Nature Pub. Group Country of Publication: United States NLM ID: 101231976 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1552-4469 (Electronic) Linking ISSN: 15524450 NLM ISO Abbreviation: Nat Chem Biol Subsets: MEDLINE

An NMDAR positive and negative allosteric modulator series share a binding site and are interconverted by methyl groups.

Authors: Perszyk R Katzman BM Kusumoto H et al.

Source: ELife [Elife] 2018 May 24; Vol. 7. Date of Electronic Publication: 2018 May 24.

Publication Type: Journal Article; Research Support, N.I.H., Extramural

Journal Info: Publisher: eLife Sciences Publications, Ltd Country of Publication: England NLM ID: 101579614 Publication Model: Electronic Cited Medium: Internet ISSN: 2050-084X (Electronic) Linking ISSN: 2050084X NLM ISO Abbreviation: Elife Subsets: MEDLINE

The Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA Receptor.

Authors: Kaiser TM Kell SA Kusumoto H et al.

Source: Molecular pharmacology [Mol Pharmacol] 2018 Feb; Vol. 93 (2), pp. 141-156. Date of Electronic Publication: 2017 Dec 14.

Publication Type: Journal Article; Research Support, N.I.H., Extramural

Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 0035623 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-0111 (Electronic) Linking ISSN: 0026895X NLM ISO Abbreviation: Mol Pharmacol Subsets: MEDLINE

The Structure-Activity Relationship of a Tetrahydroisoquinoline Class of N-Methyl-d-Aspartate Receptor Modulators that Potentiates GluN2B-Containing N-Methyl-d-Aspartate Receptors.

Authors: Strong KL Epplin MP Bacsa J et al.

Source: Journal of medicinal chemistry [J Med Chem] 2017 Jul 13; Vol. 60 (13), pp. 5556-5585. Date of Electronic Publication: 2017 Jun 26.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, N.I.H., Extramural

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE