Search Results - "Evindar G"

Author Correction: Prioritizing multiple therapeutic targets in parallel using automated DNA-encoded library screening.

Authors: Machutta CA Kollmann CS Lind KE et al.

Source: Nature communications [Nat Commun] 2018 Jul 13; Vol. 9, pp. 16227. Date of Electronic Publication: 2018 Jul 13.

Publication Type: Journal Article; Published Erratum

Journal Info: Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101528555 Publication Model: Electronic Cited Medium: Internet ISSN: 2041-1723 (Electronic) Linking ISSN: 20411723 NLM ISO Abbreviation: Nat Commun Subsets: PubMed not MEDLINE

Prioritizing multiple therapeutic targets in parallel using automated DNA-encoded library screening.

Authors: Machutta CA Kollmann CS Lind KE et al.

Source: Nature communications [Nat Commun] 2017 Jul 17; Vol. 8, pp. 16081. Date of Electronic Publication: 2017 Jul 17.

Publication Type: Journal Article

Journal Info: Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101528555 Publication Model: Electronic Cited Medium: Internet ISSN: 2041-1723 (Electronic) Linking ISSN: 20411723 NLM ISO Abbreviation: Nat Commun Subsets: MEDLINE

In Vivo Half-Life Extension of BMP1/TLL Metalloproteinase Inhibitors Using Small-Molecule Human Serum Albumin Binders.

Authors: Vantourout JC Mason AM Yuen J et al.

Source: Bioconjugate chemistry [Bioconjug Chem] 2021 Feb 17; Vol. 32 (2), pp. 279-289. Date of Electronic Publication: 2021 Feb 01.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9010319 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4812 (Electronic) Linking ISSN: 10431802 NLM ISO Abbreviation: Bioconjug Chem Subsets: MEDLINE

DNA-Encoded Library Technology-Based Discovery, Lead Optimization, and Prodrug Strategy toward Structurally Unique Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors.

Authors: Kazmierski WM Xia B Miller J et al.

Source: Journal of medicinal chemistry [J Med Chem] 2020 Apr 09; Vol. 63 (7), pp. 3552-3562. Date of Electronic Publication: 2020 Mar 19.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Development of a Selection Method for Discovering Irreversible (Covalent) Binders from a DNA-Encoded Library.

Authors: Zhu Z Grady LC Ding Y et al.

Source: SLAS discovery : advancing life sciences R & D [SLAS Discov] 2019 Feb; Vol. 24 (2), pp. 169-174. Date of Electronic Publication: 2018 Nov 01.

Publication Type: Journal Article

Journal Info: Publisher: SAGE Publications Country of Publication: United States NLM ID: 101697563 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2472-5560 (Electronic) Linking ISSN: 24725552 NLM ISO Abbreviation: SLAS Discov Subsets: MEDLINE

Design and Application of a DNA-Encoded Macrocyclic Peptide Library.

Authors: Zhu Z Shaginian A Grady LC et al.

Source: ACS chemical biology [ACS Chem Biol] 2018 Jan 19; Vol. 13 (1), pp. 53-59. Date of Electronic Publication: 2017 Dec 04.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE

Discovery and Characterization of a Class of Pyrazole Inhibitors of Bacterial Undecaprenyl Pyrophosphate Synthase.

Authors: Concha N Huang J Bai X et al.

Source: Journal of medicinal chemistry [J Med Chem] 2016 Aug 11; Vol. 59 (15), pp. 7299-304. Date of Electronic Publication: 2016 Jul 20.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Discovery of a Potent Class of PI3Kα Inhibitors with Unique Binding Mode via Encoded Library Technology (ELT).

Authors: Yang H Medeiros PF Raha K et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2015 Mar 20; Vol. 6 (5), pp. 531-6. Date of Electronic Publication: 2015 Mar 20 (Print Publication: 2015).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Application of encoded library technology (ELT) to a protein-protein interaction target: discovery of a potent class of integrin lymphocyte function-associated antigen 1 (LFA-1) antagonists.

Authors: Kollmann CS Bai X Tsai CH et al.

Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2014 Apr 01; Vol. 22 (7), pp. 2353-65. Date of Electronic Publication: 2014 Feb 07.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE

Encoded library technology as a source of hits for the discovery and lead optimization of a potent and selective class of bactericidal direct inhibitors of Mycobacterium tuberculosis InhA.

Authors: Encinas L O'Keefe H Neu M et al.

Source: Journal of medicinal chemistry [J Med Chem] 2014 Feb 27; Vol. 57 (4), pp. 1276-88. Date of Electronic Publication: 2014 Feb 05.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.

Authors: Deng H Bernier SG Doyle E et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2013 Aug 27; Vol. 4 (10), pp. 942-7. Date of Electronic Publication: 2013 Aug 27 (Print Publication: 2013).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Discovery of thieno[3,2-d]pyrimidine-6-carboxamides as potent inhibitors of SIRT1, SIRT2, and SIRT3.

Authors: Disch JS Evindar G Chiu CH et al.

Source: Journal of medicinal chemistry [J Med Chem] 2013 May 09; Vol. 56 (9), pp. 3666-79. Date of Electronic Publication: 2013 Apr 29.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Exploring amino acids derivatives as potent, selective, and direct agonists of sphingosine-1-phosphate receptor subtype-1.

Authors: Evindar G Deng H Bernier SG et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2013 Jan 15; Vol. 23 (2), pp. 472-5. Date of Electronic Publication: 2012 Nov 27.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

The Discovery of VX-745: A Novel and Selective p38α Kinase Inhibitor.

Authors: Duffy JP Harrington EM Salituro FG et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2011 Jul 28; Vol. 2 (10), pp. 758-63. Date of Electronic Publication: 2011 Jul 28 (Print Publication: 2011).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Exploration of amino alcohol derivatives as novel, potent, and highly selective sphingosine-1-phosphate receptor subtype-1 agonists.

Authors: Evindar G Bernier SG Doyle E et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2010 Apr 15; Vol. 20 (8), pp. 2520-4. Date of Electronic Publication: 2010 Mar 03.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Synthesis and evaluation of arylalkoxy- and biarylalkoxy-phenylamide and phenylimidazoles as potent and selective sphingosine-1-phosphate receptor subtype-1 agonists.

Authors: Evindar G Satz AL Bernier SG et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2009 Apr 15; Vol. 19 (8), pp. 2315-9. Date of Electronic Publication: 2009 Feb 23.

Publication Type: Comparative Study; Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Synthesis and evaluation of alkoxy-phenylamides and alkoxy-phenylimidazoles as potent sphingosine-1-phosphate receptor subtype-1 agonists.

Authors: Evindar G Bernier SG Kavarana MJ et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2009 Jan 15; Vol. 19 (2), pp. 369-72. Date of Electronic Publication: 2008 Nov 24.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Copper-catalyzed domino annulation approaches to the synthesis of benzoxazoles under microwave-accelerated and conventional thermal conditions.

Authors: Viirre RD Evindar G Batey RA

Source: The Journal of organic chemistry [J Org Chem] 2008 May 02; Vol. 73 (9), pp. 3452-9. Date of Electronic Publication: 2008 Apr 01.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 2985193R Publication Model: Print-Electronic Cited Medium: Print ISSN: 0022-3263 (Print) Linking ISSN: 00223263 NLM ISO Abbreviation: J Org Chem Subsets: MEDLINE

Peptide-heterocycle hybrid molecules: solid-phase-supported synthesis of substituted N-terminal 5-aminotetrazole peptides via electrocyclization of peptidic imidoylazides.

Authors: Gavrilyuk JI Evindar G Chen JY et al.

Source: Journal of combinatorial chemistry [J Comb Chem] 2007 Jul-Aug; Vol. 9 (4), pp. 644-51. Date of Electronic Publication: 2007 Jun 20.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 100886263 Publication Model: Print-Electronic Cited Medium: Print ISSN: 1520-4766 (Print) Linking ISSN: 15204766 NLM ISO Abbreviation: J Comb Chem Subsets: MEDLINE

Parallel synthesis of a library of benzoxazoles and benzothiazoles using ligand-accelerated copper-catalyzed cyclizations of ortho-halobenzanilides.

Authors: Evindar G Batey RA

Source: The Journal of organic chemistry [J Org Chem] 2006 Mar 03; Vol. 71 (5), pp. 1802-8.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 2985193R Publication Model: Print Cited Medium: Print ISSN: 0022-3263 (Print) Linking ISSN: 00223263 NLM ISO Abbreviation: J Org Chem Subsets: MEDLINE