Search Results - "GABA agonists"

Design, Synthesis, Biological Evaluation, and Computational Studies of Novel 1,4-Diketopiperazines as GABA Agonist.

Authors: Anwar MAE Mohammed ER El Moghazy SM et al.

Source: Drug development research [Drug Dev Res] 2025 Aug; Vol. 86 (5), pp. e70136.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-Liss Country of Publication: United States NLM ID: 8204468 Publication Model: Print Cited Medium: Internet ISSN: 1098-2299 (Electronic) Linking ISSN: 02724391 NLM ISO Abbreviation: Drug Dev Res Subsets: MEDLINE

Null method to estimate the maximal PA at subsaturating concentrations of agonist.

Authors: Germann AL Pierce SR Steinbach JH et al.

Source: The Journal of general physiology [J Gen Physiol] 2025 Jan 06; Vol. 157 (1). Date of Electronic Publication: 2024 Nov 25.

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Rockefeller University Press Country of Publication: United States NLM ID: 2985110R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1540-7748 (Electronic) Linking ISSN: 00221295 NLM ISO Abbreviation: J Gen Physiol Subsets: MEDLINE

GABA Receptor Activation in Müller Glia as a Molecular Switch for Controlling VEGF-A in the Retina.

Authors: Medina-Arellano AE Albert-Garay JS Tovar-Hernandez K et al.

Source: ASN neuro [ASN Neuro] 2026 Jan 28; Vol. 18 (1), pp. 2618997. Date of Electronic Publication: 2026 Feb 01.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Taylor & Francis Country of Publication: United States NLM ID: 101507115 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1759-0914 (Electronic) Linking ISSN: 17590914 NLM ISO Abbreviation: ASN Neuro Subsets: MEDLINE

Use of Both Fluoro-Jade B and Hematoxylin and Eosin to Detect Cell Death in the Juvenile Rat Brain Exposed to NMDA-Receptor Antagonists or GABA-Receptor Agonists in Safety Assessment.

Authors: Picut CA Mendes OR Weil DS et al.

Source: Toxicologic pathology [Toxicol Pathol] 2021 Jul; Vol. 49 (5), pp. 1109-1116. Date of Electronic Publication: 2021 Jun 02.

Publication Type: Journal Article

Journal Info: Publisher: Sage Publications Country of Publication: United States NLM ID: 7905907 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1533-1601 (Electronic) Linking ISSN: 01926233 NLM ISO Abbreviation: Toxicol Pathol Subsets: MEDLINE

Sexual behavior, lipid peroxidation and androgenic function in adult rats following pubertate stress: effects of a GABA agonist or vitamin E.

Alternate Title: СТАТЕВА ПОВЕДІНКА, ПЕРЕКИСНЕ ОКИСНЕННЯ ЛІПІДІВ І АНДРОГЕННА ФУНКЦІЯ У ДОРОСЛИХ ЩУРІВ ПІСЛЯ ПУБЕРТАТНОГО СТРЕСУ НА ТЛІ ЗАСТОСУВАННЯ АГОНІСТА ГАМК АБО ВІТАМІНУ Е.

Authors: Reznikov, A. G. Lymareva, A. A. Sachynska, O. V. et al.

Source: Physiological Journal / Fiziologichnyi Zhurnal. 2025, Vol. 71 Issue 4, p3-10. 8p.

Recurrent neonatal seizures increase tonic inhibition and respond to enhancers of δ-containing GABAA receptors.

Authors: Liddiard GT Buchanan GF Schultz ML et al.

Source: JCI insight [JCI Insight] 2025 Sep 16; Vol. 10 (21). Date of Electronic Publication: 2025 Sep 16 (Print Publication: 2025).

Publication Type: Journal Article

Journal Info: Publisher: American Society for Clinical Investigation Country of Publication: United States NLM ID: 101676073 Publication Model: eCollection Cited Medium: Internet ISSN: 2379-3708 (Electronic) Linking ISSN: 23793708 NLM ISO Abbreviation: JCI Insight Subsets: MEDLINE

Muscimol-induced inactivation of the anterior cingulate cortex does not impair trace fear conditioning in the rat.

Authors: Pezze MA Marshall HJ Cassaday HJ

Source: Journal of psychopharmacology (Oxford, England) [J Psychopharmacol] 2020 Dec; Vol. 34 (12), pp. 1457-1460. Date of Electronic Publication: 2020 Nov 08.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Sage Publications Country of Publication: United States NLM ID: 8907828 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1461-7285 (Electronic) Linking ISSN: 02698811 NLM ISO Abbreviation: J Psychopharmacol Subsets: MEDLINE

Dissociable contributions of mediodorsal and anterior thalamic nuclei in visual attentional performance: A comparison using nicotinic and muscarinic cholinergic receptor antagonists.

Authors: Mantanona CP Božič T Chudasama Y et al.

Source: Journal of psychopharmacology (Oxford, England) [J Psychopharmacol] 2020 Dec; Vol. 34 (12), pp. 1371-1381. Date of Electronic Publication: 2020 Oct 24.

Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Intramural; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Sage Publications Country of Publication: United States NLM ID: 8907828 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1461-7285 (Electronic) Linking ISSN: 02698811 NLM ISO Abbreviation: J Psychopharmacol Subsets: MEDLINE

Efficient Generation of Megakaryocyte Progenitors and Platelets From HSPCs via JAK2/STAT3 Signaling.

Authors: Liu, Huicong Wang, Lingna Liu, Jiaqing et al.

Source: Advanced Science. 6/20/2025, Vol. 12 Issue 23, p1-14. 14p.

GABA and astrocytic cholesterol determine the lipid environment of GABAAR in cultured cortical neurons.

Authors: Yuan, Zixuan Pavel, Mahmud Arif Hansen, Scott B.

Source: Communications Biology. 4/22/2025, Vol. 8 Issue 1, p1-13. 13p.

Antiepileptic Activity of Callicarpa kwangtungensis Chun Extract in Pilocarpine Induced Epilepsy in Mice via Modulating GABAergic and DAergic Transmission.

Authors: Shiqing Li Meizhi Li Rutong Wei et al.

Source: BioResources. 2025, Vol. 20 Issue 2, p4701-4719. 19p.

Exploring new cyclohexane carboxamides based GABA agonist: Design, synthesis, biological evaluation, in silico ADME and docking studies.

Authors: Hamada Abd-Allah W Abd El-Mohsen Anwar M Mohammed ER et al.

Source: Bioorganic chemistry [Bioorg Chem] 2023 Jul; Vol. 136, pp. 106561. Date of Electronic Publication: 2023 Apr 25.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

A hypothalamus-habenula circuit regulates psychomotor responses induced by cocaine.

Authors: Ahn DB Jang HB Ryu Y et al.

Source: Addiction biology [Addict Biol] 2023 Dec; Vol. 28 (12), pp. e13354.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-Blackwell Country of Publication: United States NLM ID: 9604935 Publication Model: Print Cited Medium: Internet ISSN: 1369-1600 (Electronic) Linking ISSN: 13556215 NLM ISO Abbreviation: Addict Biol Subsets: MEDLINE

Design, Synthesis, Anticonvulsant Evaluation, and Molecular Docking Studies of New GABAA Agonist Derivatives.

Authors: Koopaei, Mansur Nassiri Moghimirad, Parsa Moghadam, Ebrahim Saeedian et al.

Source: IJ Pharmaceutical Research (IJPR). Jan-Dec2025, Vol. 24 Issue 1, p1-13. 13p.

Valence-dependent contribution by the basolateral amygdala to active but not inhibitory avoidance and reward-seeking.

Authors: Dalton GL Daly ID Floresco SB

Source: Behavioural brain research [Behav Brain Res] 2025 Apr 27; Vol. 484, pp. 115503. Date of Electronic Publication: 2025 Feb 20.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier/North-Holland Biomedical Press Country of Publication: Netherlands NLM ID: 8004872 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-7549 (Electronic) Linking ISSN: 01664328 NLM ISO Abbreviation: Behav Brain Res Subsets: MEDLINE

Muscimol injection in the thalamic reticular nucleus reverts the effect of dopaminergic lesion on short-term memory in the rat globus pallidus externus.

Authors: Alexis EC Janeth MZ Daniel RJ et al.

Source: Brain research [Brain Res] 2025 Apr 01; Vol. 1852, pp. 149495. Date of Electronic Publication: 2025 Feb 07.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier/North-Holland Biomedical Press Country of Publication: Netherlands NLM ID: 0045503 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-6240 (Electronic) Linking ISSN: 00068993 NLM ISO Abbreviation: Brain Res Subsets: MEDLINE

'I haven't discussed anything with anyone': lived experience of long-term users of benzodiazepine receptor agonists regarding their treatment for substance use disorder.

Authors: Van Ngoc, Pauline Ceuterick, Melissa Belche, Jean-Luc et al.

Source: International Journal of Qualitative Studies on Health & Well-Being. Dec2024, Vol. 19 Issue 1, p1-12. 12p.

The efficacy of ciprofol versus propofol on anesthesia in patients undergoing endoscopy: a systematic review and meta-analysis of randomized controlled trials.

Authors: Liu, Jikai Hong, Aonan Zeng, Jinfang et al.

Source: BMC Anesthesiology. 10/8/2024, Vol. 24 Issue 1, p1-12. 12p.

A Withdrawal Syndrome After a Switch of Phenibut to Another γ-Aminobutyric Acid Agonist.

Authors: Pain S Bouquet E Coulon M et al.

Source: Journal of clinical psychopharmacology [J Clin Psychopharmacol] 2022 Sep-Oct 01; Vol. 42 (5), pp. 500-501. Date of Electronic Publication: 2022 Aug 06.

Publication Type: Journal Article

Journal Info: Publisher: Williams And Wilkins Country of Publication: United States NLM ID: 8109496 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1533-712X (Electronic) Linking ISSN: 02710749 NLM ISO Abbreviation: J Clin Psychopharmacol Subsets: MEDLINE

Translocator protein agonist Ro5-4864 alleviates neuropathic pain and promotes remyelination in the sciatic nerve.

Authors: Ma B Liu X Huang X et al.

Source: Molecular pain [Mol Pain] 2018 Jan-Dec; Vol. 14, pp. 1744806917748019. Date of Electronic Publication: 2017 Dec 06.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Sage Publications Inc Country of Publication: United States NLM ID: 101242662 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1744-8069 (Electronic) Linking ISSN: 17448069 NLM ISO Abbreviation: Mol Pain Subsets: MEDLINE