Search Results - "Pottie E"

TRACT assay-based in vitro characterization of substituted cathinones: inhibition and release at the serotonin transporter.

Authors: Timmerman A Pottie E Stove CP

Source: Archives of toxicology [Arch Toxicol] 2026 Jun; Vol. 100 (6), pp. 2581-2598. Date of Electronic Publication: 2026 Mar 31.

Publication Type: Journal Article

Journal Info: Publisher: Springer-Verlag Country of Publication: Germany NLM ID: 0417615 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1432-0738 (Electronic) Linking ISSN: 03405761 NLM ISO Abbreviation: Arch Toxicol Subsets: MEDLINE

In vitro bioassays for measuring monoamine transporter function.

Authors: Timmerman A Baumann M Bosmans F et al.

Source: Neuropharmacology [Neuropharmacology] 2026 May 30; Vol. 298, pp. 111053. Date of Electronic Publication: 2026 May 30.

Publication Type: Journal Article; Review

Journal Info: Publisher: Pergamon Press Country of Publication: England NLM ID: 0236217 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-7064 (Electronic) Linking ISSN: 00283908 NLM ISO Abbreviation: Neuropharmacology Subsets: MEDLINE

N‑Benzyl-Tryptamine Derivatives as Serotonin 5‑HT2 Receptor Ligands: Synthesis and Structure-Affinity/Activity Relationships.

Authors: Martínez-Afani D Soares BA Mella-Raipán J et al.

Source: ACS omega [ACS Omega] 2026 May 13; Vol. 11 (20), pp. 29638-29653. Date of Electronic Publication: 2026 May 13 (Print Publication: 2026).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101691658 Publication Model: eCollection Cited Medium: Internet ISSN: 2470-1343 (Electronic) Linking ISSN: 24701343 NLM ISO Abbreviation: ACS Omega Subsets: PubMed not MEDLINE

Pain management beyond opioids: a β-arrestin2-biased allosteric GPCR modulator opens new avenues for drug development.

Authors: Pottie E Steinmüller SAM Decker M

Source: Signal transduction and targeted therapy [Signal Transduct Target Ther] 2025 Aug 27; Vol. 10 (1), pp. 264. Date of Electronic Publication: 2025 Aug 27.

Publication Type: Journal Article

Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101676423 Publication Model: Electronic Cited Medium: Internet ISSN: 2059-3635 (Electronic) Linking ISSN: 20593635 NLM ISO Abbreviation: Signal Transduct Target Ther Subsets: MEDLINE; In Process

The psychedelic phenethylamine 25C-NBF, a selective 5-HT2A agonist, shows psychoplastogenic properties and rapid antidepressant effects in male rodents.

Authors: Nadal-Gratacós N Puigseslloses P Guzmán L et al.

Source: Molecular psychiatry [Mol Psychiatry] 2026 Apr; Vol. 31 (4), pp. 1909-1922. Date of Electronic Publication: 2025 Nov 14.

Publication Type: Journal Article

Journal Info: Publisher: Nature Publishing Group Specialist Journals Country of Publication: England NLM ID: 9607835 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5578 (Electronic) Linking ISSN: 13594184 NLM ISO Abbreviation: Mol Psychiatry Subsets: MEDLINE

N-Benzyl-tryptamine Derivatives as Serotonin 5-HT2A Receptor (5-HT2AR) Agonists: Focus on Different In Vitro 5-HT2AR Activity Profiles.

Authors: Pottie E Vertriest E Martínez-Afani D et al.

Source: ACS chemical neuroscience [ACS Chem Neurosci] 2026 Apr 01; Vol. 17 (7), pp. 1256-1268. Date of Electronic Publication: 2026 Mar 20.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101525337 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1948-7193 (Electronic) Linking ISSN: 19487193 NLM ISO Abbreviation: ACS Chem Neurosci Subsets: MEDLINE

The 4-alkyl chain length of 2,5-dimethoxyamphetamines differentially affects in vitro serotonin receptor actions versus in vivo psychedelic-like effects.

Authors: Luethi D Glatfelter GC Pottie E et al.

Source: Molecular psychiatry [Mol Psychiatry] 2026 Mar; Vol. 31 (3), pp. 1799-1809. Date of Electronic Publication: 2025 Nov 05.

Publication Type: Journal Article

Journal Info: Publisher: Nature Publishing Group Specialist Journals Country of Publication: England NLM ID: 9607835 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5578 (Electronic) Linking ISSN: 13594184 NLM ISO Abbreviation: Mol Psychiatry Subsets: MEDLINE

Neuropharmacology of halogenated DMT analogs: psychoplastogenic and antidepressant properties of 5-Br-DMT, a psychedelic derivative with low hallucinogenic potential.

Authors: Puigseslloses P Nadal-Gratacós N Fumàs B et al.

Source: Molecular psychiatry [Mol Psychiatry] 2026 Mar; Vol. 31 (3), pp. 1733-1745. Date of Electronic Publication: 2025 Oct 21.

Publication Type: Journal Article

Journal Info: Publisher: Nature Publishing Group Specialist Journals Country of Publication: England NLM ID: 9607835 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5578 (Electronic) Linking ISSN: 13594184 NLM ISO Abbreviation: Mol Psychiatry Subsets: MEDLINE

Live cell luminescence-based Gαq-PLC-β interaction assay: Development and application at the serotonin 5-HT2A receptor.

Authors: Pottie E Stove CP

Source: Pharmacological research [Pharmacol Res] 2026 Feb; Vol. 224, pp. 108094. Date of Electronic Publication: 2026 Jan 10.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 8907422 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1096-1186 (Electronic) Linking ISSN: 10436618 NLM ISO Abbreviation: Pharmacol Res Subsets: MEDLINE

In vitro structure-activity relationships and forensic case series of emerging 2-benzylbenzimidazole 'nitazene' opioids.

Authors: De Vrieze LM Walton SE Pottie E et al.

Source: Archives of toxicology [Arch Toxicol] 2024 Sep; Vol. 98 (9), pp. 2999-3018. Date of Electronic Publication: 2024 Jun 14.

Publication Type: Journal Article

Journal Info: Publisher: Springer-Verlag Country of Publication: Germany NLM ID: 0417615 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1432-0738 (Electronic) Linking ISSN: 03405761 NLM ISO Abbreviation: Arch Toxicol Subsets: MEDLINE

Activity-based detection of synthetic cannabinoid receptor agonists in plant materials.

Authors: Timmerman A Balcaen M Coopman V et al.

Source: Harm reduction journal [Harm Reduct J] 2024 Jul 01; Vol. 21 (1), pp. 127. Date of Electronic Publication: 2024 Jul 01.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: BioMed Central Country of Publication: England NLM ID: 101153624 Publication Model: Electronic Cited Medium: Internet ISSN: 1477-7517 (Electronic) Linking ISSN: 14777517 NLM ISO Abbreviation: Harm Reduct J Subsets: MEDLINE

Setup and Evaluation of the TRACT Assay Principle for the In Vitro Functional Characterization of Modulators of the Serotonin Transporter and the Serotonin 2A Receptor.

Authors: Timmerman A Walther D Baumann MH et al.

Source: Analytical chemistry [Anal Chem] 2025 Aug 19; Vol. 97 (32), pp. 17872-17881. Date of Electronic Publication: 2025 Aug 06.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 0370536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-6882 (Electronic) Linking ISSN: 00032700 NLM ISO Abbreviation: Anal Chem Subsets: MEDLINE

Design, Synthesis, and In Vitro Characterization of a Tryptamine-Based Visible-Light Photoswitchable 5-HT2AR Ligand Showing Efficacy Preference for β-Arrestin over Mini-Gq.

Authors: Sink A Pottie E Carter SJ et al.

Source: Journal of medicinal chemistry [J Med Chem] 2025 Jul 10; Vol. 68 (13), pp. 13628-13639. Date of Electronic Publication: 2025 Jun 18.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Off-target activity of NBOMes and NBOMe analogs at the µ opioid receptor.

Authors: Deventer MH Persson M Laus A et al.

Source: Archives of toxicology [Arch Toxicol] 2023 May; Vol. 97 (5), pp. 1367-1384. Date of Electronic Publication: 2023 Feb 28.

Publication Type: Journal Article

Journal Info: Publisher: Springer-Verlag Country of Publication: Germany NLM ID: 0417615 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1432-0738 (Electronic) Linking ISSN: 03405761 NLM ISO Abbreviation: Arch Toxicol Subsets: MEDLINE

Synthesis, Pharmacological Characterization, and Binding Mode Analysis of 8-Hydroxy-Tetrahydroisoquinolines as 5-HT7 Receptor Inverse Agonists.

Authors: Chan CB Pottie E Simon IA et al.

Source: ACS chemical neuroscience [ACS Chem Neurosci] 2025 Feb 05; Vol. 16 (3), pp. 439-451. Date of Electronic Publication: 2025 Jan 21.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101525337 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1948-7193 (Electronic) Linking ISSN: 19487193 NLM ISO Abbreviation: ACS Chem Neurosci Subsets: MEDLINE

In vitro assays for the functional characterization of (psychedelic) substances at the serotonin receptor 5-HT2A R.

Authors: Pottie E Stove CP

Source: Journal of neurochemistry [J Neurochem] 2022 Jul; Vol. 162 (1), pp. 39-59. Date of Electronic Publication: 2022 Jan 17.

Publication Type: Journal Article; Review

Journal Info: Publisher: Wiley on behalf of the International Society for Neurochemistry Country of Publication: England NLM ID: 2985190R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1471-4159 (Electronic) Linking ISSN: 00223042 NLM ISO Abbreviation: J Neurochem Subsets: MEDLINE

2-Substituted (N)-Methanocarba A3 Adenosine Receptor Agonists: In Silico, In Vitro, and In Vivo Characterization.

Authors: Tosh DK Pavan M Cronin C et al.

Source: ACS pharmacology & translational science [ACS Pharmacol Transl Sci] 2024 Jun 06; Vol. 7 (7), pp. 2154-2173. Date of Electronic Publication: 2024 Jun 06 (Print Publication: 2024).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101721411 Publication Model: eCollection Cited Medium: Internet ISSN: 2575-9108 (Electronic) Linking ISSN: 25759108 NLM ISO Abbreviation: ACS Pharmacol Transl Sci Subsets: PubMed not MEDLINE

Selective Replacement of Cholesterol with Cationic Amphiphilic Drugs Enables the Design of Lipid Nanoparticles with Improved RNA Delivery.

Authors: Bogaert B Debisschop A Ehouarne T et al.

Source: Nano letters [Nano Lett] 2024 Mar 13; Vol. 24 (10), pp. 2961-2971. Date of Electronic Publication: 2024 Mar 04.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101088070 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1530-6992 (Electronic) Linking ISSN: 15306984 NLM ISO Abbreviation: Nano Lett Subsets: MEDLINE

Comparative Pharmacological Effects of Lisuride and Lysergic Acid Diethylamide Revisited.

Authors: Glatfelter GC Pottie E Partilla JS et al.

Source: ACS pharmacology & translational science [ACS Pharmacol Transl Sci] 2024 Feb 05; Vol. 7 (3), pp. 641-653. Date of Electronic Publication: 2024 Feb 05 (Print Publication: 2024).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101721411 Publication Model: eCollection Cited Medium: Internet ISSN: 2575-9108 (Electronic) Linking ISSN: 25759108 NLM ISO Abbreviation: ACS Pharmacol Transl Sci Subsets: PubMed not MEDLINE

In vitro structure-activity relationship determination of 30 psychedelic new psychoactive substances by means of β-arrestin 2 recruitment to the serotonin 2A receptor.

Authors: Pottie E Cannaert A Stove CP

Source: Archives of toxicology [Arch Toxicol] 2020 Oct; Vol. 94 (10), pp. 3449-3460. Date of Electronic Publication: 2020 Jul 05.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Springer-Verlag Country of Publication: Germany NLM ID: 0417615 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1432-0738 (Electronic) Linking ISSN: 03405761 NLM ISO Abbreviation: Arch Toxicol Subsets: MEDLINE