Synthesis and biological evaluation of piperazinyl heterocyclic antagonists of the gonadotropin releasing hormone (GnRH) receptor.

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Title: Synthesis and biological evaluation of piperazinyl heterocyclic antagonists of the gonadotropin releasing hormone (GnRH) receptor.
Authors: Vera MD; Department of Chemical, Wyeth Research, Collegeville, PA 19426, USA., Lundquist JT 4th, Chengalvala MV, Cottom JE, Feingold IB, Garrick LM, Green DM, Hauze DB, Mann CW, Mehlmann JF, Rogers JF, Shanno L, Wrobel JE, Pelletier JC
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2010 Apr 15; Vol. 20 (8), pp. 2512-5. Date of Electronic Publication: 2010 Mar 03.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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DbLabel: MEDLINE Ultimate
An: 20236823
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PubType: Academic Journal
PubTypeId: academicJournal
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  Data: Synthesis and biological evaluation of piperazinyl heterocyclic antagonists of the gonadotropin releasing hormone (GnRH) receptor.
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  Data: <searchLink fieldCode="AU" term="%22Vera+MD%22">Vera MD</searchLink>; Department of Chemical, Wyeth Research, Collegeville, PA 19426, USA.<br /><searchLink fieldCode="AU" term="%22Lundquist+JT+4th%22">Lundquist JT 4th</searchLink><br /><searchLink fieldCode="AU" term="%22Chengalvala+MV%22">Chengalvala MV</searchLink><br /><searchLink fieldCode="AU" term="%22Cottom+JE%22">Cottom JE</searchLink><br /><searchLink fieldCode="AU" term="%22Feingold+IB%22">Feingold IB</searchLink><br /><searchLink fieldCode="AU" term="%22Garrick+LM%22">Garrick LM</searchLink><br /><searchLink fieldCode="AU" term="%22Green+DM%22">Green DM</searchLink><br /><searchLink fieldCode="AU" term="%22Hauze+DB%22">Hauze DB</searchLink><br /><searchLink fieldCode="AU" term="%22Mann+CW%22">Mann CW</searchLink><br /><searchLink fieldCode="AU" term="%22Mehlmann+JF%22">Mehlmann JF</searchLink><br /><searchLink fieldCode="AU" term="%22Rogers+JF%22">Rogers JF</searchLink><br /><searchLink fieldCode="AU" term="%22Shanno+L%22">Shanno L</searchLink><br /><searchLink fieldCode="AU" term="%22Wrobel+JE%22">Wrobel JE</searchLink><br /><searchLink fieldCode="AU" term="%22Pelletier+JC%22">Pelletier JC</searchLink>
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  Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2010 Apr 15; Vol. 20 (8), pp. 2512-5. <i>Date of Electronic Publication: </i>2010 Mar 03.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE
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        Value: 10.1016/j.bmcl.2010.02.099
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              Text: 2010 Apr 15
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