Diazepam Promotes Translocation of Human Constitutive Androstane Receptor (CAR) via Direct Interaction with the Ligand-Binding Domain.

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Title: Diazepam Promotes Translocation of Human Constitutive Androstane Receptor (CAR) via Direct Interaction with the Ligand-Binding Domain.
Authors: Skoda J; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic., Dusek J; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic., Drastik M; Department of Physical Chemistry and Biophysics, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic., Stefela A; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic., Dohnalova K; 1st Medical Faculty, Charles University, Katerinská 32, 121 08 Prague, Czech Republic.; Czech Centre for Phenogenomics, Institute of Molecular Genetics of the Czech Academy of Sciences, Vídeňská 1083, 142 20 Prague, Czech Republic., Chalupsky K; Czech Centre for Phenogenomics, Institute of Molecular Genetics of the Czech Academy of Sciences, Vídeňská 1083, 142 20 Prague, Czech Republic., Smutny T; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic., Micuda S; Department of Pharmacology, Medical Faculty in Hradec Kralove, Charles University, Simkova 870, 500 03 Hradec Kralove, Czech Republic., Gerbal-Chaloin S; IRMB, University of Montpellier, INSERM, 34295 Montpellier, France., Pavek P; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic.
Source: Cells [Cells] 2020 Nov 24; Vol. 9 (12). Date of Electronic Publication: 2020 Nov 24.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101600052 Publication Model: Electronic Cited Medium: Internet ISSN: 2073-4409 (Electronic) Linking ISSN: 20734409 NLM ISO Abbreviation: Cells Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Diazepam Promotes Translocation of Human Constitutive Androstane Receptor (CAR) via Direct Interaction with the Ligand-Binding Domain.
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  Data: <searchLink fieldCode="AU" term="%22Skoda+J%22">Skoda J</searchLink>; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Dusek+J%22">Dusek J</searchLink>; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Drastik+M%22">Drastik M</searchLink>; Department of Physical Chemistry and Biophysics, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Stefela+A%22">Stefela A</searchLink>; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Dohnalova+K%22">Dohnalova K</searchLink>; 1st Medical Faculty, Charles University, Katerinská 32, 121 08 Prague, Czech Republic.; Czech Centre for Phenogenomics, Institute of Molecular Genetics of the Czech Academy of Sciences, Vídeňská 1083, 142 20 Prague, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Chalupsky+K%22">Chalupsky K</searchLink>; Czech Centre for Phenogenomics, Institute of Molecular Genetics of the Czech Academy of Sciences, Vídeňská 1083, 142 20 Prague, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Smutny+T%22">Smutny T</searchLink>; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Micuda+S%22">Micuda S</searchLink>; Department of Pharmacology, Medical Faculty in Hradec Kralove, Charles University, Simkova 870, 500 03 Hradec Kralove, Czech Republic.<br /><searchLink fieldCode="AU" term="%22Gerbal-Chaloin+S%22">Gerbal-Chaloin S</searchLink>; IRMB, University of Montpellier, INSERM, 34295 Montpellier, France.<br /><searchLink fieldCode="AU" term="%22Pavek+P%22">Pavek P</searchLink>; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Charles University, Heyrovskeho 1203, 500 05 Hradec Kralove, Czech Republic.
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  Data: <searchLink fieldCode="JN" term="%22101600052%22">Cells</searchLink> [Cells] 2020 Nov 24; Vol. 9 (12). <i>Date of Electronic Publication: </i>2020 Nov 24.
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              Text: 2020 Nov 24
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