In Vivo Half-Life Extension of BMP1/TLL Metalloproteinase Inhibitors Using Small-Molecule Human Serum Albumin Binders.

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Title: In Vivo Half-Life Extension of BMP1/TLL Metalloproteinase Inhibitors Using Small-Molecule Human Serum Albumin Binders.
Authors: Vantourout JC; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K.; Department of Pure and Applied Chemistry, University of Strathclyde, 295 Cathedral Street, Glasgow G11XL, U.K., Mason AM; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Yuen J; GlaxoSmithKline US, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States., Simpson GL; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Evindar G; GlaxoSmithKline US, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States., Kuai L; GlaxoSmithKline US, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States., Hobbs M; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Edgar E; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Needle S; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Bai X; GlaxoSmithKline US, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States., Wilson S; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Scott-Stevens P; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Traylen W; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Lambert K; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Young N; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Bunally S; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Summerfield SG; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Snell R; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Lad R; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Shi E; GlaxoSmithKline US, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States., Skinner S; GlaxoSmithKline US, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States., Shewchuk L; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Watson AJB; University of St Andrews, North Haugh, St Andrews KY16 9ST, U.K., Chung CW; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Pal S; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K., Holt DA; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Kallander LS; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Prendergast J; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Rivera K; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Washburn DG; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Harpel MR; GlaxoSmithKline US, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, United States., Arico-Muendel C; GlaxoSmithKline US, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States., Isidro-Llobet A; GlaxoSmithKline U.K., Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K.
Source: Bioconjugate chemistry [Bioconjug Chem] 2021 Feb 17; Vol. 32 (2), pp. 279-289. Date of Electronic Publication: 2021 Feb 01.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9010319 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4812 (Electronic) Linking ISSN: 10431802 NLM ISO Abbreviation: Bioconjug Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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