4-Substituted Thieno[3,2-d]pyrimidines as Dual-Stage Antiplasmodial Derivatives.

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Title: 4-Substituted Thieno[3,2-d]pyrimidines as Dual-Stage Antiplasmodial Derivatives.
Authors: Lagardère P; Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, UFR des Sciences Pharmaceutiques et Biologiques, 34293 Montpellier, France., Mustière R; Aix Marseille Univ, CNRS, ICR UMR 7273, Equipe Pharmaco-Chimie Radicalaire, Faculté de Pharmacie, 13385 Marseille, France., Amanzougaghene N; Centre d'Immunologie et des Maladies Infectieuses (CIMI), INSERM, CNRS, Sorbonne Université, 75013 Paris, France., Hutter S; Aix Marseille Univ, IRD, AP-HM, SSA, VITROME, 13005 Marseille, France., Franetich JF; Centre d'Immunologie et des Maladies Infectieuses (CIMI), INSERM, CNRS, Sorbonne Université, 75013 Paris, France., Azas N; Aix Marseille Univ, IRD, AP-HM, SSA, VITROME, 13005 Marseille, France., Vanelle P; Aix Marseille Univ, CNRS, ICR UMR 7273, Equipe Pharmaco-Chimie Radicalaire, Faculté de Pharmacie, 13385 Marseille, France.; Service Central de la Qualité et de l'Information Pharmaceutiques, AP-HM, Hôpital Conception, 13005 Marseille, France., Verhaeghe P; CHU de Nîmes, Service de Pharmacie, 30029 Nîmes, France.; LCC-CNRS, Université de Toulouse, CNRS UPR 8241, UPS, 31400 Toulouse, France., Primas N; Aix Marseille Univ, CNRS, ICR UMR 7273, Equipe Pharmaco-Chimie Radicalaire, Faculté de Pharmacie, 13385 Marseille, France.; Service Central de la Qualité et de l'Information Pharmaceutiques, AP-HM, Hôpital Conception, 13005 Marseille, France., Mazier D; Centre d'Immunologie et des Maladies Infectieuses (CIMI), INSERM, CNRS, Sorbonne Université, 75013 Paris, France., Masurier N; Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, UFR des Sciences Pharmaceutiques et Biologiques, 34293 Montpellier, France., Lisowski V; Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, UFR des Sciences Pharmaceutiques et Biologiques, 34293 Montpellier, France.
Source: Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2022 Jul 01; Vol. 15 (7). Date of Electronic Publication: 2022 Jul 01.
Publication Type: Journal Article
Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101238453 Publication Model: Electronic Cited Medium: Print ISSN: 1424-8247 (Print) Linking ISSN: 14248247 NLM ISO Abbreviation: Pharmaceuticals (Basel) Subsets: PubMed not MEDLINE
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  Data: 4-Substituted Thieno[3,2-d]pyrimidines as Dual-Stage Antiplasmodial Derivatives.
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  Data: <searchLink fieldCode="AU" term="%22Lagardère+P%22">Lagardère P</searchLink>; Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, UFR des Sciences Pharmaceutiques et Biologiques, 34293 Montpellier, France.<br /><searchLink fieldCode="AU" term="%22Mustière+R%22">Mustière R</searchLink>; Aix Marseille Univ, CNRS, ICR UMR 7273, Equipe Pharmaco-Chimie Radicalaire, Faculté de Pharmacie, 13385 Marseille, France.<br /><searchLink fieldCode="AU" term="%22Amanzougaghene+N%22">Amanzougaghene N</searchLink>; Centre d'Immunologie et des Maladies Infectieuses (CIMI), INSERM, CNRS, Sorbonne Université, 75013 Paris, France.<br /><searchLink fieldCode="AU" term="%22Hutter+S%22">Hutter S</searchLink>; Aix Marseille Univ, IRD, AP-HM, SSA, VITROME, 13005 Marseille, France.<br /><searchLink fieldCode="AU" term="%22Franetich+JF%22">Franetich JF</searchLink>; Centre d'Immunologie et des Maladies Infectieuses (CIMI), INSERM, CNRS, Sorbonne Université, 75013 Paris, France.<br /><searchLink fieldCode="AU" term="%22Azas+N%22">Azas N</searchLink>; Aix Marseille Univ, IRD, AP-HM, SSA, VITROME, 13005 Marseille, France.<br /><searchLink fieldCode="AU" term="%22Vanelle+P%22">Vanelle P</searchLink>; Aix Marseille Univ, CNRS, ICR UMR 7273, Equipe Pharmaco-Chimie Radicalaire, Faculté de Pharmacie, 13385 Marseille, France.; Service Central de la Qualité et de l'Information Pharmaceutiques, AP-HM, Hôpital Conception, 13005 Marseille, France.<br /><searchLink fieldCode="AU" term="%22Verhaeghe+P%22">Verhaeghe P</searchLink>; CHU de Nîmes, Service de Pharmacie, 30029 Nîmes, France.; LCC-CNRS, Université de Toulouse, CNRS UPR 8241, UPS, 31400 Toulouse, France.<br /><searchLink fieldCode="AU" term="%22Primas+N%22">Primas N</searchLink>; Aix Marseille Univ, CNRS, ICR UMR 7273, Equipe Pharmaco-Chimie Radicalaire, Faculté de Pharmacie, 13385 Marseille, France.; Service Central de la Qualité et de l'Information Pharmaceutiques, AP-HM, Hôpital Conception, 13005 Marseille, France.<br /><searchLink fieldCode="AU" term="%22Mazier+D%22">Mazier D</searchLink>; Centre d'Immunologie et des Maladies Infectieuses (CIMI), INSERM, CNRS, Sorbonne Université, 75013 Paris, France.<br /><searchLink fieldCode="AU" term="%22Masurier+N%22">Masurier N</searchLink>; Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, UFR des Sciences Pharmaceutiques et Biologiques, 34293 Montpellier, France.<br /><searchLink fieldCode="AU" term="%22Lisowski+V%22">Lisowski V</searchLink>; Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, UFR des Sciences Pharmaceutiques et Biologiques, 34293 Montpellier, France.
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