Small Molecule BRD4 Inhibitors Apabetalone and JQ1 Rescues Endothelial Cells Dysfunction, Protects Monolayer Integrity and Reduces Midkine Expression.

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Title: Small Molecule BRD4 Inhibitors Apabetalone and JQ1 Rescues Endothelial Cells Dysfunction, Protects Monolayer Integrity and Reduces Midkine Expression.
Authors: Shahid S; Institute for Clinical Chemistry, University Medical Centre Goettingen, 37075 Goettingen, Germany., Pantakani M; Institute for Clinical Chemistry, University Medical Centre Goettingen, 37075 Goettingen, Germany., Binder L; Institute for Clinical Chemistry, University Medical Centre Goettingen, 37075 Goettingen, Germany.; German Centre for Cardiovascular Research (DZHK), Partner Site Goettingen, 37075 Goettingen, Germany., Fischer A; Institute for Clinical Chemistry, University Medical Centre Goettingen, 37075 Goettingen, Germany.; German Centre for Cardiovascular Research (DZHK), Partner Site Goettingen, 37075 Goettingen, Germany.; Division Vascular Signaling and Cancer, German Cancer Research Center (DKFZ), 69120 Heidelberg, Germany., Pantakani K; Institute for Clinical Chemistry, University Medical Centre Goettingen, 37075 Goettingen, Germany.; German Centre for Cardiovascular Research (DZHK), Partner Site Goettingen, 37075 Goettingen, Germany., Asif AR; Institute for Clinical Chemistry, University Medical Centre Goettingen, 37075 Goettingen, Germany.; German Centre for Cardiovascular Research (DZHK), Partner Site Goettingen, 37075 Goettingen, Germany.
Source: Molecules (Basel, Switzerland) [Molecules] 2022 Nov 02; Vol. 27 (21). Date of Electronic Publication: 2022 Nov 02.
Publication Type: Journal Article
Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1420-3049
DOI:10.3390/molecules27217453