Evaluation of the Gly-Phe-Lys Linker to Reduce the Renal Radioactivity of a [64Cu]Cu-Labeled Multimeric cRGD Peptide.

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Title: Evaluation of the Gly-Phe-Lys Linker to Reduce the Renal Radioactivity of a [64Cu]Cu-Labeled Multimeric cRGD Peptide.
Authors: Jin ZH; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Degardin M; Département de Chimie Moléculaire, CNRS, Université Grenoble Alpes, cedex 9, Grenoble 38058, France., Furukawa T; Department of Integrated Health Sciences, Graduate School of Medicine, Nagoya University, Nagoya 461-8673, Japan.; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Uehara T; Laboratory of Molecular Imaging and Radiotherapy, Graduate School of Pharmaceutical Sciences, Chiba University, Chiba 260-8675, Japan., Tsuji AB; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Suzuki H; Laboratory of Molecular Imaging and Radiotherapy, Graduate School of Pharmaceutical Sciences, Chiba University, Chiba 260-8675, Japan., Wakizaka H; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Sugyo A; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Aung W; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Suzuki H; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Nagatsu K; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Zhang MR; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan., Dumy P; Institut des Biomolécules Max Mousseron, École Nationale Supérieure de Chimie de Montpellier, Université de Montpellier, cedex 5, Montpellier 34296, France., Boturyn D; Département de Chimie Moléculaire, CNRS, Université Grenoble Alpes, cedex 9, Grenoble 38058, France., Higashi T; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.
Source: ACS omega [ACS Omega] 2025 Jan 24; Vol. 10 (4), pp. 4102-4120. Date of Electronic Publication: 2025 Jan 24 (Print Publication: 2025).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101691658 Publication Model: eCollection Cited Medium: Internet ISSN: 2470-1343 (Electronic) Linking ISSN: 24701343 NLM ISO Abbreviation: ACS Omega Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: Evaluation of the Gly-Phe-Lys Linker to Reduce the Renal Radioactivity of a [<superscript>64</superscript>Cu]Cu-Labeled Multimeric cRGD Peptide.
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  Data: <searchLink fieldCode="AU" term="%22Jin+ZH%22">Jin ZH</searchLink>; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Degardin+M%22">Degardin M</searchLink>; Département de Chimie Moléculaire, CNRS, Université Grenoble Alpes, cedex 9, Grenoble 38058, France.<br /><searchLink fieldCode="AU" term="%22Furukawa+T%22">Furukawa T</searchLink>; Department of Integrated Health Sciences, Graduate School of Medicine, Nagoya University, Nagoya 461-8673, Japan.; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Uehara+T%22">Uehara T</searchLink>; Laboratory of Molecular Imaging and Radiotherapy, Graduate School of Pharmaceutical Sciences, Chiba University, Chiba 260-8675, Japan.<br /><searchLink fieldCode="AU" term="%22Tsuji+AB%22">Tsuji AB</searchLink>; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Suzuki+H%22">Suzuki H</searchLink>; Laboratory of Molecular Imaging and Radiotherapy, Graduate School of Pharmaceutical Sciences, Chiba University, Chiba 260-8675, Japan.<br /><searchLink fieldCode="AU" term="%22Wakizaka+H%22">Wakizaka H</searchLink>; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Sugyo+A%22">Sugyo A</searchLink>; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Aung+W%22">Aung W</searchLink>; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Suzuki+H%22">Suzuki H</searchLink>; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Nagatsu+K%22">Nagatsu K</searchLink>; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Zhang+MR%22">Zhang MR</searchLink>; Department of Advanced Nuclear Medicine Sciences, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.<br /><searchLink fieldCode="AU" term="%22Dumy+P%22">Dumy P</searchLink>; Institut des Biomolécules Max Mousseron, École Nationale Supérieure de Chimie de Montpellier, Université de Montpellier, cedex 5, Montpellier 34296, France.<br /><searchLink fieldCode="AU" term="%22Boturyn+D%22">Boturyn D</searchLink>; Département de Chimie Moléculaire, CNRS, Université Grenoble Alpes, cedex 9, Grenoble 38058, France.<br /><searchLink fieldCode="AU" term="%22Higashi+T%22">Higashi T</searchLink>; Department of Molecular Imaging and Theranostics, Institute for Quantum Medical Science, National Institutes for Quantum Science and Technology (QST), Chiba 263-8555, Japan.
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