In Vitro and In Vivo Pharmacokinetic Characterization of 7-Hydroxymitragynine, an Active Metabolite of Mitragynine, in Sprague-Dawley Rats.
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| Title: | In Vitro and In Vivo Pharmacokinetic Characterization of 7-Hydroxymitragynine, an Active Metabolite of Mitragynine, in Sprague-Dawley Rats. |
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| Authors: | Chiang YH; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA., Kanumuri SRR; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA.; Translational Drug Development Core, Clinical and Translational Science Institute, University of Florida, Gainesville, FL, USA., Kuntz MA; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA., Senetra AS; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA., Berthold EC; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA., Kamble SH; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA., Mukhopadhyay S; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, FL, USA., Hampson AJ; Division of Therapeutics and Medical Consequences, National Institute on Drug Abuse, National Institutes of Health, Bethesda, MD, USA., McCurdy CR; Translational Drug Development Core, Clinical and Translational Science Institute, University of Florida, Gainesville, FL, USA.; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, FL, USA., Sharma A; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA. asharma1@cop.ufl.edu.; Translational Drug Development Core, Clinical and Translational Science Institute, University of Florida, Gainesville, FL, USA. asharma1@cop.ufl.edu. |
| Source: | European journal of drug metabolism and pharmacokinetics [Eur J Drug Metab Pharmacokinet] 2025 May; Vol. 50 (3), pp. 205-218. Date of Electronic Publication: 2025 Mar 22. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Springer France Country of Publication: France NLM ID: 7608491 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2107-0180 (Electronic) Linking ISSN: 03787966 NLM ISO Abbreviation: Eur J Drug Metab Pharmacokinet Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 40119246 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: In Vitro and In Vivo Pharmacokinetic Characterization of 7-Hydroxymitragynine, an Active Metabolite of Mitragynine, in Sprague-Dawley Rats. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Chiang+YH%22">Chiang YH</searchLink>; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA.<br /><searchLink fieldCode="AU" term="%22Kanumuri+SRR%22">Kanumuri SRR</searchLink>; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA.; Translational Drug Development Core, Clinical and Translational Science Institute, University of Florida, Gainesville, FL, USA.<br /><searchLink fieldCode="AU" term="%22Kuntz+MA%22">Kuntz MA</searchLink>; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA.<br /><searchLink fieldCode="AU" term="%22Senetra+AS%22">Senetra AS</searchLink>; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA.<br /><searchLink fieldCode="AU" term="%22Berthold+EC%22">Berthold EC</searchLink>; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA.<br /><searchLink fieldCode="AU" term="%22Kamble+SH%22">Kamble SH</searchLink>; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA.<br /><searchLink fieldCode="AU" term="%22Mukhopadhyay+S%22">Mukhopadhyay S</searchLink>; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, FL, USA.<br /><searchLink fieldCode="AU" term="%22Hampson+AJ%22">Hampson AJ</searchLink>; Division of Therapeutics and Medical Consequences, National Institute on Drug Abuse, National Institutes of Health, Bethesda, MD, USA.<br /><searchLink fieldCode="AU" term="%22McCurdy+CR%22">McCurdy CR</searchLink>; Translational Drug Development Core, Clinical and Translational Science Institute, University of Florida, Gainesville, FL, USA.; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, FL, USA.<br /><searchLink fieldCode="AU" term="%22Sharma+A%22">Sharma A</searchLink>; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive Medical Sciences Building MSB P3-20B, Gainesville, FL, 32610, USA. asharma1@cop.ufl.edu.; Translational Drug Development Core, Clinical and Translational Science Institute, University of Florida, Gainesville, FL, USA. asharma1@cop.ufl.edu. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%227608491%22">European journal of drug metabolism and pharmacokinetics</searchLink> [Eur J Drug Metab Pharmacokinet] 2025 May; Vol. 50 (3), pp. 205-218. <i>Date of Electronic Publication: </i>2025 Mar 22. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Springer+France%22">Springer France </searchLink><i>Country of Publication: </i>France <i>NLM ID: </i>7608491 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2107-0180 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2203787966%22">03787966 </searchLink><i>NLM ISO Abbreviation: </i>Eur J Drug Metab Pharmacokinet <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=40119246 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1007/s13318-025-00939-2 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 205 Titles: – TitleFull: In Vitro and In Vivo Pharmacokinetic Characterization of 7-Hydroxymitragynine, an Active Metabolite of Mitragynine, in Sprague-Dawley Rats. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Chiang YH – PersonEntity: Name: NameFull: Kanumuri SRR – PersonEntity: Name: NameFull: Kuntz MA – PersonEntity: Name: NameFull: Senetra AS – PersonEntity: Name: NameFull: Berthold EC – PersonEntity: Name: NameFull: Kamble SH – PersonEntity: Name: NameFull: Mukhopadhyay S – PersonEntity: Name: NameFull: Hampson AJ – PersonEntity: Name: NameFull: McCurdy CR – PersonEntity: Name: NameFull: Sharma A IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 05 Text: 2025 May Type: published Y: 2025 Identifiers: – Type: issn-electronic Value: 2107-0180 Numbering: – Type: volume Value: 50 – Type: issue Value: 3 Titles: – TitleFull: European journal of drug metabolism and pharmacokinetics Type: main |
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