Novel Potent and Selective Dopamine D4 Receptor Piperidine Antagonists as Potential Alternatives for the Treatment of Glioblastoma.

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Title: Novel Potent and Selective Dopamine D4 Receptor Piperidine Antagonists as Potential Alternatives for the Treatment of Glioblastoma.
Authors: Matteucci F; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Pavletić P; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.; Faculty of Biotechnology and Drug Development, University of Rijeka, 51000 Rijeka, Croatia., Bonifazi A; Department of Pharmacology and Toxicology, Center for Addiction Sciences and Therapeutics, University of Texas Medical Branch, Galveston, TX 77555, USA., Garland R; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA., Yano H; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA., Amantini C; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy., Zeppa L; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy., Sabato E; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy., Vistoli G; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy., Mammoli V; Center for Drug Discovery and Development-IDD, Aptuit, an Evotec Company, 37135 Verona, Italy., Cappellacci L; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Del Bello F; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Giorgioni G; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Petrelli R; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Piergentili A; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Quaglia W; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Piergentili A; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.
Source: Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2025 May 17; Vol. 18 (5). Date of Electronic Publication: 2025 May 17.
Publication Type: Journal Article
Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101238453 Publication Model: Electronic Cited Medium: Print ISSN: 1424-8247 (Print) Linking ISSN: 14248247 NLM ISO Abbreviation: Pharmaceuticals (Basel) Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: Novel Potent and Selective Dopamine D4 Receptor Piperidine Antagonists as Potential Alternatives for the Treatment of Glioblastoma.
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  Data: <searchLink fieldCode="AU" term="%22Matteucci+F%22">Matteucci F</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Pavletić+P%22">Pavletić P</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.; Faculty of Biotechnology and Drug Development, University of Rijeka, 51000 Rijeka, Croatia.<br /><searchLink fieldCode="AU" term="%22Bonifazi+A%22">Bonifazi A</searchLink>; Department of Pharmacology and Toxicology, Center for Addiction Sciences and Therapeutics, University of Texas Medical Branch, Galveston, TX 77555, USA.<br /><searchLink fieldCode="AU" term="%22Garland+R%22">Garland R</searchLink>; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA.<br /><searchLink fieldCode="AU" term="%22Yano+H%22">Yano H</searchLink>; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA.<br /><searchLink fieldCode="AU" term="%22Amantini+C%22">Amantini C</searchLink>; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Zeppa+L%22">Zeppa L</searchLink>; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Sabato+E%22">Sabato E</searchLink>; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy.<br /><searchLink fieldCode="AU" term="%22Vistoli+G%22">Vistoli G</searchLink>; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy.<br /><searchLink fieldCode="AU" term="%22Mammoli+V%22">Mammoli V</searchLink>; Center for Drug Discovery and Development-IDD, Aptuit, an Evotec Company, 37135 Verona, Italy.<br /><searchLink fieldCode="AU" term="%22Cappellacci+L%22">Cappellacci L</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Del+Bello+F%22">Del Bello F</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Giorgioni+G%22">Giorgioni G</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Petrelli+R%22">Petrelli R</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Piergentili+A%22">Piergentili A</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Quaglia+W%22">Quaglia W</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Piergentili+A%22">Piergentili A</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.
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