Novel Potent and Selective Dopamine D4 Receptor Piperidine Antagonists as Potential Alternatives for the Treatment of Glioblastoma.
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| Title: | Novel Potent and Selective Dopamine D4 Receptor Piperidine Antagonists as Potential Alternatives for the Treatment of Glioblastoma. |
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| Authors: | Matteucci F; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Pavletić P; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.; Faculty of Biotechnology and Drug Development, University of Rijeka, 51000 Rijeka, Croatia., Bonifazi A; Department of Pharmacology and Toxicology, Center for Addiction Sciences and Therapeutics, University of Texas Medical Branch, Galveston, TX 77555, USA., Garland R; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA., Yano H; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA., Amantini C; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy., Zeppa L; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy., Sabato E; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy., Vistoli G; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy., Mammoli V; Center for Drug Discovery and Development-IDD, Aptuit, an Evotec Company, 37135 Verona, Italy., Cappellacci L; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Del Bello F; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Giorgioni G; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Petrelli R; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Piergentili A; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Quaglia W; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy., Piergentili A; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy. |
| Source: | Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2025 May 17; Vol. 18 (5). Date of Electronic Publication: 2025 May 17. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: MDPI Country of Publication: Switzerland NLM ID: 101238453 Publication Model: Electronic Cited Medium: Print ISSN: 1424-8247 (Print) Linking ISSN: 14248247 NLM ISO Abbreviation: Pharmaceuticals (Basel) Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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| FullText | Links: – Type: pdflink Text: Availability: 1 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 40430557 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Novel Potent and Selective Dopamine D4 Receptor Piperidine Antagonists as Potential Alternatives for the Treatment of Glioblastoma. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Matteucci+F%22">Matteucci F</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Pavletić+P%22">Pavletić P</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.; Faculty of Biotechnology and Drug Development, University of Rijeka, 51000 Rijeka, Croatia.<br /><searchLink fieldCode="AU" term="%22Bonifazi+A%22">Bonifazi A</searchLink>; Department of Pharmacology and Toxicology, Center for Addiction Sciences and Therapeutics, University of Texas Medical Branch, Galveston, TX 77555, USA.<br /><searchLink fieldCode="AU" term="%22Garland+R%22">Garland R</searchLink>; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA.<br /><searchLink fieldCode="AU" term="%22Yano+H%22">Yano H</searchLink>; Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, MA 02115, USA.<br /><searchLink fieldCode="AU" term="%22Amantini+C%22">Amantini C</searchLink>; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Zeppa+L%22">Zeppa L</searchLink>; Immunopathology and Molecular Medicine Unit, School of Biosciences and Veterinary Medicine, University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Sabato+E%22">Sabato E</searchLink>; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy.<br /><searchLink fieldCode="AU" term="%22Vistoli+G%22">Vistoli G</searchLink>; Department of Pharmaceutical Sciences, University of Milan, 20133 Milano, Italy.<br /><searchLink fieldCode="AU" term="%22Mammoli+V%22">Mammoli V</searchLink>; Center for Drug Discovery and Development-IDD, Aptuit, an Evotec Company, 37135 Verona, Italy.<br /><searchLink fieldCode="AU" term="%22Cappellacci+L%22">Cappellacci L</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Del+Bello+F%22">Del Bello F</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Giorgioni+G%22">Giorgioni G</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Petrelli+R%22">Petrelli R</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Piergentili+A%22">Piergentili A</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Quaglia+W%22">Quaglia W</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy.<br /><searchLink fieldCode="AU" term="%22Piergentili+A%22">Piergentili A</searchLink>; Medicinal Chemistry Unit, School of Pharmacy, Chemistry Interdisciplinary Project (ChIP), University of Camerino, 62032 Camerino, Italy. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101238453%22">Pharmaceuticals (Basel, Switzerland)</searchLink> [Pharmaceuticals (Basel)] 2025 May 17; Vol. 18 (5). <i>Date of Electronic Publication: </i>2025 May 17. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22MDPI%22">MDPI </searchLink><i>Country of Publication: </i>Switzerland <i>NLM ID: </i>101238453 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Print <i>ISSN: </i>1424-8247 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2214248247%22">14248247 </searchLink><i>NLM ISO Abbreviation: </i>Pharmaceuticals (Basel) <i>Subsets: </i>PubMed not MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=40430557 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.3390/ph18050739 Languages: – Code: eng Text: English Titles: – TitleFull: Novel Potent and Selective Dopamine D4 Receptor Piperidine Antagonists as Potential Alternatives for the Treatment of Glioblastoma. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Matteucci F – PersonEntity: Name: NameFull: Pavletić P – PersonEntity: Name: NameFull: Bonifazi A – PersonEntity: Name: NameFull: Garland R – PersonEntity: Name: NameFull: Yano H – PersonEntity: Name: NameFull: Amantini C – PersonEntity: Name: NameFull: Zeppa L – PersonEntity: Name: NameFull: Sabato E – PersonEntity: Name: NameFull: Vistoli G – PersonEntity: Name: NameFull: Mammoli V – PersonEntity: Name: NameFull: Cappellacci L – PersonEntity: Name: NameFull: Del Bello F – PersonEntity: Name: NameFull: Giorgioni G – PersonEntity: Name: NameFull: Petrelli R – PersonEntity: Name: NameFull: Piergentili A – PersonEntity: Name: NameFull: Quaglia W – PersonEntity: Name: NameFull: Piergentili A IsPartOfRelationships: – BibEntity: Dates: – D: 17 M: 05 Text: 2025 May 17 Type: published Y: 2025 Identifiers: – Type: issn-print Value: 1424-8247 Numbering: – Type: volume Value: 18 – Type: issue Value: 5 Titles: – TitleFull: Pharmaceuticals (Basel, Switzerland) Type: main |
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