Novel indole-based indoleamine 2,3-dioxygenase-1 (IDO1) inhibitors: design, synthesis, and antidepressant evaluation.
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| Title: | Novel indole-based indoleamine 2,3-dioxygenase-1 (IDO1) inhibitors: design, synthesis, and antidepressant evaluation. |
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| Authors: | Zhang J; School of Biological Science and Technology, University of Jinan, Jinan 250022, China., Gao WJ; Shandong Laboratory of Yantai Drug Discovery, Bohai Rim Advanced Research Institute for Drug Discovery, Yantai, Shandong 264117, China., Zheng YX; School of Biological Science and Technology, University of Jinan, Jinan 250022, China., Shao JD; Advanced Medical Research Institute, Cheeloo College of Medicine, Shandong University, Jinan, Shandong 250012, China., Zhang NY; School of Biological Science and Technology, University of Jinan, Jinan 250022, China., Guo W; School of Biological Science and Technology, University of Jinan, Jinan 250022, China., Wang S; School of Biological Science and Technology, University of Jinan, Jinan 250022, China., Zhao Q; Cambrian Neuroscience Inc., No. 3-1, Xinjinhu Road, Jiangbei New District, Nanjing 210032, China., Zhu K; Advanced Medical Research Institute, Cheeloo College of Medicine, Shandong University, Jinan, Shandong 250012, China.; The Second Hospital of Shandong University, Cheeloo College of Medicine, Shandong University, Jinan, Shandong 250012, China.. Electronic address: hkhhh.k@163.com., Gao M; Cambrian Neuroscience Inc., No. 3-1, Xinjinhu Road, Jiangbei New District, Nanjing 210032, China. Electronic address: gaoming@cambrian-ns.com., Yu JH; Shandong Laboratory of Yantai Drug Discovery, Bohai Rim Advanced Research Institute for Drug Discovery, Yantai, Shandong 264117, China. Electronic address: jhyu@baridd.ac.cn., Meng N; School of Biological Science and Technology, University of Jinan, Jinan 250022, China. Electronic address: mls_mengn@ujn.edu.cn., Jiang CS; School of Biological Science and Technology, University of Jinan, Jinan 250022, China. Electronic address: bio_jiangcs@ujn.edu.cn. |
| Source: | Bioorganic & medicinal chemistry [Bioorg Med Chem] 2026 Feb; Vol. 133, pp. 118503. Date of Electronic Publication: 2025 Dec 02. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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