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Development of indole derived non-orthosteric inhibitors for Proto-oncogene serine/threonine-protein kinase PIM-1.

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Title: Development of indole derived non-orthosteric inhibitors for Proto-oncogene serine/threonine-protein kinase PIM-1.
Authors: Grau BW; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA., Tailor D; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA., Pandrala M; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA., Schultz KJ; Computational Biology Group, Pacific Northwest National Laboratory, Richland, WA, 99354, USA., Hsu EC; Department of Radiology, Canary Center at Stanford for Cancer Early Detection, Stanford University School of Medicine, Palo Alto, CA, 94304, USA., Dheeraj A; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA., Rolig AS; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA., Struntz NB; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA., Luong P; Department of Biomolecular Systems, Max-Planck-Institute of Colloids and Interfaces, Am Mühlenberg 1, Potsdam-Golm, 14476, Germany; Bowdoin College, 6600 College Station, Brunswick, ME, 04011, USA., Stoyanova T; Department of Radiology, Canary Center at Stanford for Cancer Early Detection, Stanford University School of Medicine, Palo Alto, CA, 94304, USA., Sledge GW; Department of Medicine, Stanford University School of Medicine, Palo Alto, CA, 94304, USA; Stanford Cancer Institute, Stanford University School of Medicine, Stanford, CA, 94305, USA., Malhotra SV; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA. Electronic address: malhotsa@ohsu.edu.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2026 May 29; Vol. 316, pp. 118931. Date of Electronic Publication: 2026 May 29.
Publication Type: Journal Article
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
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  Data: Development of indole derived non-orthosteric inhibitors for Proto-oncogene serine/threonine-protein kinase PIM-1.
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  Data: <searchLink fieldCode="AU" term="%22Grau+BW%22">Grau BW</searchLink>; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA.<br /><searchLink fieldCode="AU" term="%22Tailor+D%22">Tailor D</searchLink>; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA.<br /><searchLink fieldCode="AU" term="%22Pandrala+M%22">Pandrala M</searchLink>; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA.<br /><searchLink fieldCode="AU" term="%22Schultz+KJ%22">Schultz KJ</searchLink>; Computational Biology Group, Pacific Northwest National Laboratory, Richland, WA, 99354, USA.<br /><searchLink fieldCode="AU" term="%22Hsu+EC%22">Hsu EC</searchLink>; Department of Radiology, Canary Center at Stanford for Cancer Early Detection, Stanford University School of Medicine, Palo Alto, CA, 94304, USA.<br /><searchLink fieldCode="AU" term="%22Dheeraj+A%22">Dheeraj A</searchLink>; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA.<br /><searchLink fieldCode="AU" term="%22Rolig+AS%22">Rolig AS</searchLink>; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA.<br /><searchLink fieldCode="AU" term="%22Struntz+NB%22">Struntz NB</searchLink>; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA.<br /><searchLink fieldCode="AU" term="%22Luong+P%22">Luong P</searchLink>; Department of Biomolecular Systems, Max-Planck-Institute of Colloids and Interfaces, Am Mühlenberg 1, Potsdam-Golm, 14476, Germany; Bowdoin College, 6600 College Station, Brunswick, ME, 04011, USA.<br /><searchLink fieldCode="AU" term="%22Stoyanova+T%22">Stoyanova T</searchLink>; Department of Radiology, Canary Center at Stanford for Cancer Early Detection, Stanford University School of Medicine, Palo Alto, CA, 94304, USA.<br /><searchLink fieldCode="AU" term="%22Sledge+GW%22">Sledge GW</searchLink>; Department of Medicine, Stanford University School of Medicine, Palo Alto, CA, 94304, USA; Stanford Cancer Institute, Stanford University School of Medicine, Stanford, CA, 94305, USA.<br /><searchLink fieldCode="AU" term="%22Malhotra+SV%22">Malhotra SV</searchLink>; Department of Cell, Development and Cancer Biology, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA; Center for Experimental Therapeutics, Knight Cancer Institute, Oregon Health & Science University, Portland, OR, 97239, USA. Electronic address: malhotsa@ohsu.edu.
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  Data: <searchLink fieldCode="JN" term="%220420510%22">European journal of medicinal chemistry</searchLink> [Eur J Med Chem] 2026 May 29; Vol. 316, pp. 118931. <i>Date of Electronic Publication: </i>2026 May 29.
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