Streamlined Radiosynthesis of [ 18 F]Fluproxadine (AF78): An Unprotected Guanidine Precursor Enables Efficient One-Step, Automation-Ready Labeling for Clinical Use.

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Title: Streamlined Radiosynthesis of [ 18 F]Fluproxadine (AF78): An Unprotected Guanidine Precursor Enables Efficient One-Step, Automation-Ready Labeling for Clinical Use.
Authors: Chen, Xinyu1 (AUTHOR), Ohta, Kaito2,3 (AUTHOR), Kimura, Hiroyuki3,4 (AUTHOR), Yagi, Yusuke3,4,5 (AUTHOR), Sasaki, Takanori3,5 (AUTHOR), Nose, Naoko3,6 (AUTHOR), Akehi, Masaru3,7 (AUTHOR), Yamane, Tomohiko6,8 (AUTHOR), Werner, Rudolf A.1,7,8 (AUTHOR), Higuchi, Takahiro2,3 (AUTHOR) thiguchi@me.com
Source: Pharmaceutics. Jan2026, Vol. 18 Issue 1, p123. 18p.
Database: Academic Search Ultimate
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ISSN:19994923
DOI:10.3390/pharmaceutics18010123