Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.

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Bibliographic Details
Title: Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.
Authors: Deng H; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Bernier SG; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Doyle E; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Lorusso J; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Morgan BA; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Westlin WF; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Evindar G; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2013 Aug 27; Vol. 4 (10), pp. 942-7. Date of Electronic Publication: 2013 Aug 27 (Print Publication: 2013).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1948-5875
DOI:10.1021/ml400194r