Benzoxaborole Antimalarial Agents. Part 5. Lead Optimization of Novel Amide Pyrazinyloxy Benzoxaboroles and Identification of a Preclinical Candidate.
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| Title: | Benzoxaborole Antimalarial Agents. Part 5. Lead Optimization of Novel Amide Pyrazinyloxy Benzoxaboroles and Identification of a Preclinical Candidate. |
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| Authors: | Zhang YK; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Plattner JJ; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Easom EE; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Jacobs RT; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Guo D; Department of Medicine, University of California, San Francisco , Box 0811, San Francisco, California 94143, United States., Freund YR; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Berry P; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Ciaravino V; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Erve JCL; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States., Rosenthal PJ; Department of Medicine, University of California, San Francisco , Box 0811, San Francisco, California 94143, United States., Campo B; Medicines for Malaria Venture, International Center Cointrin , Block G, 20 Route de Pré-Bois, POB 1826, CH - 1215 Geneva, Switzerland., Gamo FJ; Diseases of the Developing World, GlaxoSmithKline , Severo Ochoa 2, 28760, Tres Cantos, Spain., Sanz LM; Diseases of the Developing World, GlaxoSmithKline , Severo Ochoa 2, 28760, Tres Cantos, Spain., Cao J; Shanghai ChemPartner , 998 Ha-lei Road, Zhangjiang High-tech Park, Pudong New Area, Shanghai 201203, China. |
| Source: | Journal of medicinal chemistry [J Med Chem] 2017 Jul 13; Vol. 60 (13), pp. 5889-5908. Date of Electronic Publication: 2017 Jun 29. |
| Publication Type: | Journal Article; Research Support, N.I.H., Extramural |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 28635296 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Benzoxaborole Antimalarial Agents. Part 5. Lead Optimization of Novel Amide Pyrazinyloxy Benzoxaboroles and Identification of a Preclinical Candidate. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Zhang+YK%22">Zhang YK</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Plattner+JJ%22">Plattner JJ</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Easom+EE%22">Easom EE</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Jacobs+RT%22">Jacobs RT</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Guo+D%22">Guo D</searchLink>; Department of Medicine, University of California, San Francisco , Box 0811, San Francisco, California 94143, United States.<br /><searchLink fieldCode="AU" term="%22Freund+YR%22">Freund YR</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Berry+P%22">Berry P</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Ciaravino+V%22">Ciaravino V</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Erve+JCL%22">Erve JCL</searchLink>; Anacor Pharmaceuticals, Inc. , 1020 E. Meadow Circle, Palo Alto, California 94303, United States.<br /><searchLink fieldCode="AU" term="%22Rosenthal+PJ%22">Rosenthal PJ</searchLink>; Department of Medicine, University of California, San Francisco , Box 0811, San Francisco, California 94143, United States.<br /><searchLink fieldCode="AU" term="%22Campo+B%22">Campo B</searchLink>; Medicines for Malaria Venture, International Center Cointrin , Block G, 20 Route de Pré-Bois, POB 1826, CH - 1215 Geneva, Switzerland.<br /><searchLink fieldCode="AU" term="%22Gamo+FJ%22">Gamo FJ</searchLink>; Diseases of the Developing World, GlaxoSmithKline , Severo Ochoa 2, 28760, Tres Cantos, Spain.<br /><searchLink fieldCode="AU" term="%22Sanz+LM%22">Sanz LM</searchLink>; Diseases of the Developing World, GlaxoSmithKline , Severo Ochoa 2, 28760, Tres Cantos, Spain.<br /><searchLink fieldCode="AU" term="%22Cao+J%22">Cao J</searchLink>; Shanghai ChemPartner , 998 Ha-lei Road, Zhangjiang High-tech Park, Pudong New Area, Shanghai 201203, China. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2017 Jul 13; Vol. 60 (13), pp. 5889-5908. <i>Date of Electronic Publication: </i>2017 Jun 29. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, N.I.H., Extramural – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=28635296 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acs.jmedchem.7b00621 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 5889 Titles: – TitleFull: Benzoxaborole Antimalarial Agents. Part 5. Lead Optimization of Novel Amide Pyrazinyloxy Benzoxaboroles and Identification of a Preclinical Candidate. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Zhang YK – PersonEntity: Name: NameFull: Plattner JJ – PersonEntity: Name: NameFull: Easom EE – PersonEntity: Name: NameFull: Jacobs RT – PersonEntity: Name: NameFull: Guo D – PersonEntity: Name: NameFull: Freund YR – PersonEntity: Name: NameFull: Berry P – PersonEntity: Name: NameFull: Ciaravino V – PersonEntity: Name: NameFull: Erve JCL – PersonEntity: Name: NameFull: Rosenthal PJ – PersonEntity: Name: NameFull: Campo B – PersonEntity: Name: NameFull: Gamo FJ – PersonEntity: Name: NameFull: Sanz LM – PersonEntity: Name: NameFull: Cao J IsPartOfRelationships: – BibEntity: Dates: – D: 13 M: 07 Text: 2017 Jul 13 Type: published Y: 2017 Identifiers: – Type: issn-electronic Value: 1520-4804 Numbering: – Type: volume Value: 60 – Type: issue Value: 13 Titles: – TitleFull: Journal of medicinal chemistry Type: main |
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