Cytochrome P450/ABC transporter inhibition simultaneously enhances ivermectin pharmacokinetics in the mammal host and pharmacodynamics in Anopheles gambiae.

Saved in:
Bibliographic Details
Title: Cytochrome P450/ABC transporter inhibition simultaneously enhances ivermectin pharmacokinetics in the mammal host and pharmacodynamics in Anopheles gambiae.
Authors: Chaccour CJ; Instituto de Salud Tropical, Universidad de Navarra, Pamplona, 31008, Spain. carlos.chaccour@isglobal.org.; ISGlobal, Barcelona Ctr. Int. Health Res. (CRESIB), Hospital Clínic - Universitat de Barcelona, Barcelona, 08036, Spain. carlos.chaccour@isglobal.org.; Centro de Investigação em Saúde de Manhiça, Maputo, 1929, Mozambique. carlos.chaccour@isglobal.org., Hammann F; Division of Clinical Pharmacology and Toxicology, University Hospital Basel and University of Basel, Basel, 4056, Switzerland., Alustiza M; Faculty of Medicine, Universidad de Navarra, Pamplona, 31008, Spain., Castejon S; Department of Microbiology, Clínica Universidad de Navarra, Pamplona, 31008, Spain., Tarimo BB; Ifakara Health Institute, Bagamoyo, Pwani, P.O. Box 74, United Republic of Tanzania., Abizanda G; Centro de Investigación Médica Aplicada, Pamplona, 31008, Spain., Irigoyen Barrio Á; Drug Development Unit Universidad de Navarra (DDUNAV), Pamplona, 31008, Spain., Martí Soler H; ISGlobal, Barcelona Ctr. Int. Health Res. (CRESIB), Hospital Clínic - Universitat de Barcelona, Barcelona, 08036, Spain., Moncada R; Department of Anaesthesia, Clínica Universidad de Navarra, Pamplona, 31008, Spain., Bilbao JI; Department of Radiology, Clínica Universidad de Navarra, Pamplona, 31008, Spain., Aldaz A; Department of Pharmacy, Clínica Universidad de Navarra, Pamplona, 31008, Spain., Maia M; Ifakara Health Institute, Bagamoyo, Pwani, P.O. Box 74, United Republic of Tanzania.; Swiss Tropical and Public Health Institute, Basel, 4051, Switzerland.; University of Basel, Basel, 4003, Switzerland.; KEMRI-Wellcome Trust Research Programme, Kilifi, Kenya., Del Pozo JL; Department of Microbiology, Clínica Universidad de Navarra, Pamplona, 31008, Spain.; Infectious Diseases Division, Clínica Universidad de Navarra, Pamplona, 31008, Spain.
Source: Scientific reports [Sci Rep] 2017 Aug 17; Vol. 7 (1), pp. 8535. Date of Electronic Publication: 2017 Aug 17.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN: 2045-2322 (Electronic) Linking ISSN: 20452322 NLM ISO Abbreviation: Sci Rep Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2045-2322
DOI:10.1038/s41598-017-08906-x