Bromodomain-Selective BET Inhibitors Are Potent Antitumor Agents against MYC-Driven Pediatric Cancer.

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Title: Bromodomain-Selective BET Inhibitors Are Potent Antitumor Agents against MYC-Driven Pediatric Cancer.
Authors: Slavish PJ; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Chi L; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Yun MK; Department of Structural Biology, St. Jude Children's Research Hospital, Memphis, Tennessee., Tsurkan L; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Martinez NE; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Jonchere B; Department of Tumor Cell Biology, St. Jude Children's Research Hospital, Memphis, Tennessee., Chai SC; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Connelly M; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Waddell MB; Molecular Interaction Analysis Shared Resource, St. Jude Children's Research Hospital, Memphis, Tennessee., Das S; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Neale G; Hartwell Center, St. Jude Children's Research Hospital, Memphis, Tennessee., Li Z; Department of Structural Biology, St. Jude Children's Research Hospital, Memphis, Tennessee., Shadrick WR; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Olsen RR; Department of Oncology, St. Jude Children's Research Hospital, Memphis, Tennessee., Freeman KW; Department of Oncology, St. Jude Children's Research Hospital, Memphis, Tennessee., Low JA; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Price JE; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Young BM; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Bharatham N; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Boyd VA; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Yang J; Department of Surgery, St. Jude Children's Research Hospital, Memphis, Tennessee., Lee RE; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Morfouace M; Department of Tumor Cell Biology, St. Jude Children's Research Hospital, Memphis, Tennessee., Roussel MF; Department of Tumor Cell Biology, St. Jude Children's Research Hospital, Memphis, Tennessee., Chen T; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., Savic D; Department of Pharmaceutical Sciences, St. Jude Children's Research Hospital, Memphis, Tennessee., Guy RK; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee., White SW; Department of Structural Biology, St. Jude Children's Research Hospital, Memphis, Tennessee., Shelat AA; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee. phil.potter@stjude.org anang.shelat@stjude.org., Potter PM; Department of Chemical Biology and Therapeutics, St. Jude Children's Research Hospital, Memphis, Tennessee. phil.potter@stjude.org anang.shelat@stjude.org.
Source: Cancer research [Cancer Res] 2020 Sep 01; Vol. 80 (17), pp. 3507-3518. Date of Electronic Publication: 2020 Jul 10.
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Association for Cancer Research Country of Publication: United States NLM ID: 2984705R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1538-7445 (Electronic) Linking ISSN: 00085472 NLM ISO Abbreviation: Cancer Res Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1538-7445
DOI:10.1158/0008-5472.CAN-19-3934