Analogues of Natural Chalcones as Efficient Inhibitors of AKR1C3.
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| Title: | Analogues of Natural Chalcones as Efficient Inhibitors of AKR1C3. |
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| Authors: | Möller G; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany., Temml V; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Cala Peralta A; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Gruet O; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Richomme P; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Séraphin D; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Viault G; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Kraus L; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Huber-Cantonati P; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Schopfhauser E; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Pachmayr J; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Tokarz J; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany., Schuster D; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Helesbeux JJ; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Dyar KA; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany. |
| Source: | Metabolites [Metabolites] 2022 Jan 21; Vol. 12 (2). Date of Electronic Publication: 2022 Jan 21. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: MDPI Country of Publication: Switzerland NLM ID: 101578790 Publication Model: Electronic Cited Medium: Print ISSN: 2218-1989 (Print) Linking ISSN: 22181989 NLM ISO Abbreviation: Metabolites Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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| ISSN: | 2218-1989 |
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| DOI: | 10.3390/metabo12020099 |