Analogues of Natural Chalcones as Efficient Inhibitors of AKR1C3.
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| Title: | Analogues of Natural Chalcones as Efficient Inhibitors of AKR1C3. |
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| Authors: | Möller G; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany., Temml V; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Cala Peralta A; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Gruet O; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Richomme P; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Séraphin D; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Viault G; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Kraus L; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Huber-Cantonati P; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Schopfhauser E; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Pachmayr J; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Tokarz J; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany., Schuster D; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria., Helesbeux JJ; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France., Dyar KA; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany. |
| Source: | Metabolites [Metabolites] 2022 Jan 21; Vol. 12 (2). Date of Electronic Publication: 2022 Jan 21. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: MDPI Country of Publication: Switzerland NLM ID: 101578790 Publication Model: Electronic Cited Medium: Print ISSN: 2218-1989 (Print) Linking ISSN: 22181989 NLM ISO Abbreviation: Metabolites Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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| FullText | Links: – Type: pdflink Text: Availability: 1 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 35208174 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Analogues of Natural Chalcones as Efficient Inhibitors of AKR1C3. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Möller+G%22">Möller G</searchLink>; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany.<br /><searchLink fieldCode="AU" term="%22Temml+V%22">Temml V</searchLink>; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria.<br /><searchLink fieldCode="AU" term="%22Cala+Peralta+A%22">Cala Peralta A</searchLink>; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France.<br /><searchLink fieldCode="AU" term="%22Gruet+O%22">Gruet O</searchLink>; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France.<br /><searchLink fieldCode="AU" term="%22Richomme+P%22">Richomme P</searchLink>; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France.<br /><searchLink fieldCode="AU" term="%22Séraphin+D%22">Séraphin D</searchLink>; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France.<br /><searchLink fieldCode="AU" term="%22Viault+G%22">Viault G</searchLink>; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France.<br /><searchLink fieldCode="AU" term="%22Kraus+L%22">Kraus L</searchLink>; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria.<br /><searchLink fieldCode="AU" term="%22Huber-Cantonati+P%22">Huber-Cantonati P</searchLink>; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria.<br /><searchLink fieldCode="AU" term="%22Schopfhauser+E%22">Schopfhauser E</searchLink>; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria.<br /><searchLink fieldCode="AU" term="%22Pachmayr+J%22">Pachmayr J</searchLink>; Institute of Pharmacy, Pharmaceutical Biology and Clinical Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria.<br /><searchLink fieldCode="AU" term="%22Tokarz+J%22">Tokarz J</searchLink>; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany.<br /><searchLink fieldCode="AU" term="%22Schuster+D%22">Schuster D</searchLink>; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University Salzburg, 5020 Salzburg, Austria.<br /><searchLink fieldCode="AU" term="%22Helesbeux+JJ%22">Helesbeux JJ</searchLink>; University of Angers, SONAS, SFR QUASAV, F-49000 Angers, France.<br /><searchLink fieldCode="AU" term="%22Dyar+KA%22">Dyar KA</searchLink>; Institute for Diabetes and Cancer, Helmholtz Center Munich, German Research Center for Environmental Health, 85764 Neuherberg, Germany. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101578790%22">Metabolites</searchLink> [Metabolites] 2022 Jan 21; Vol. 12 (2). <i>Date of Electronic Publication: </i>2022 Jan 21. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22MDPI%22">MDPI </searchLink><i>Country of Publication: </i>Switzerland <i>NLM ID: </i>101578790 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Print <i>ISSN: </i>2218-1989 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2222181989%22">22181989 </searchLink><i>NLM ISO Abbreviation: </i>Metabolites <i>Subsets: </i>PubMed not MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=35208174 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.3390/metabo12020099 Languages: – Code: eng Text: English Titles: – TitleFull: Analogues of Natural Chalcones as Efficient Inhibitors of AKR1C3. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Möller G – PersonEntity: Name: NameFull: Temml V – PersonEntity: Name: NameFull: Cala Peralta A – PersonEntity: Name: NameFull: Gruet O – PersonEntity: Name: NameFull: Richomme P – PersonEntity: Name: NameFull: Séraphin D – PersonEntity: Name: NameFull: Viault G – PersonEntity: Name: NameFull: Kraus L – PersonEntity: Name: NameFull: Huber-Cantonati P – PersonEntity: Name: NameFull: Schopfhauser E – PersonEntity: Name: NameFull: Pachmayr J – PersonEntity: Name: NameFull: Tokarz J – PersonEntity: Name: NameFull: Schuster D – PersonEntity: Name: NameFull: Helesbeux JJ – PersonEntity: Name: NameFull: Dyar KA IsPartOfRelationships: – BibEntity: Dates: – D: 21 M: 01 Text: 2022 Jan 21 Type: published Y: 2022 Identifiers: – Type: issn-print Value: 2218-1989 Numbering: – Type: volume Value: 12 – Type: issue Value: 2 Titles: – TitleFull: Metabolites Type: main |
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