Irreversible inhibition of TRF2TRFH recruiting functions by a covalent cyclic peptide induces telomeric replication stress in cancer cells.

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Title: Irreversible inhibition of TRF2TRFH recruiting functions by a covalent cyclic peptide induces telomeric replication stress in cancer cells.
Authors: Sobinoff AP; Telomere Length Regulation Unit, Children's Medical Research Institute, Faculty of Medicine and Health, University of Sydney, Westmead, NSW 2145, Australia., Di Maro S; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Low RRJ; Genome Integrity Unit, Children's Medical Research Institute, Faculty of Medicine and Health, University of Sydney, Westmead, NSW 2145, Australia., Benedetti R; Department of Precision Medicine, University of Campania 'Luigi Vanvitelli', Vico L. De Crecchio 7, 80138 Naples, Italy; Azienda Ospedaliera Universitaria 'Luigi Vanvitelli', Medical Epigenetics Program., Tomassi S; Department of Pharmacy, University of Naples 'Federico II', Via D. Montesano 49, 80131 Naples, Italy., D'Aniello A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Russo R; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Baglivo I; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Chianese U; Department of Precision Medicine, University of Campania 'Luigi Vanvitelli', Vico L. De Crecchio 7, 80138 Naples, Italy., Pedone PV; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Chambery A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Cesare AJ; Genome Integrity Unit, Children's Medical Research Institute, Faculty of Medicine and Health, University of Sydney, Westmead, NSW 2145, Australia., Altucci L; Department of Precision Medicine, University of Campania 'Luigi Vanvitelli', Vico L. De Crecchio 7, 80138 Naples, Italy; BIOGEM, 83031 Ariano Irpino, Italy; Azienda Ospedaliera Universitaria 'Luigi Vanvitelli', Medical Epigenetics Program; IEOS CNR, Napoli, Italy., Pickett HA; Telomere Length Regulation Unit, Children's Medical Research Institute, Faculty of Medicine and Health, University of Sydney, Westmead, NSW 2145, Australia. Electronic address: hpickett@cmri.org.au., Cosconati S; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy. Electronic address: sandro.cosconati@unicampania.it.
Source: Cell chemical biology [Cell Chem Biol] 2023 Dec 21; Vol. 30 (12), pp. 1652-1665.e6. Date of Electronic Publication: 2023 Dec 07.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Cell Press Country of Publication: United States NLM ID: 101676030 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2451-9448 (Electronic) Linking ISSN: 24519448 NLM ISO Abbreviation: Cell Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2451-9448
DOI:10.1016/j.chembiol.2023.11.008