AMG 193, a Clinical Stage MTA-Cooperative PRMT5 Inhibitor, Drives Antitumor Activity Preclinically and in Patients with MTAP-Deleted Cancers.

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Title: AMG 193, a Clinical Stage MTA-Cooperative PRMT5 Inhibitor, Drives Antitumor Activity Preclinically and in Patients with MTAP-Deleted Cancers.
Authors: Belmontes B; Amgen Research, Thousand Oaks, California., Slemmons KK; Amgen Research, Thousand Oaks, California., Su C; Amgen Research, South San Francisco, California., Liu S; Amgen Research, Thousand Oaks, California., Policheni AN; Amgen Research, Thousand Oaks, California., Moriguchi J; Amgen Research, Thousand Oaks, California., Tan H; Amgen Research, Thousand Oaks, California., Xie F; Amgen Research, South San Francisco, California., Aiello DA; Amgen Research, Thousand Oaks, California., Yang Y; Amgen Research, Thousand Oaks, California., Lazaro R; Amgen Research, Thousand Oaks, California., Aeffner F; Amgen Research, South San Francisco, California., Rees MG; Broad Institute of MIT and Harvard, Cambridge, Massachusetts., Ronan MM; Broad Institute of MIT and Harvard, Cambridge, Massachusetts., Roth JA; Broad Institute of MIT and Harvard, Cambridge, Massachusetts., Vestergaard M; Amgen Research, Copenhagen, Denmark., Cowland S; Amgen Research, Copenhagen, Denmark., Andersson J; Amgen Research, Copenhagen, Denmark., Sarvary I; Amgen Research, Copenhagen, Denmark., Chen Q; Amgen Research, Thousand Oaks, California., Sharma P; Amgen Research, Thousand Oaks, California., Lopez P; Amgen Research, Thousand Oaks, California., Tamayo N; Amgen Research, Thousand Oaks, California., Pettus LH; Amgen Research, Thousand Oaks, California., Ghimire-Rijal S; Amgen Research, Thousand Oaks, California., Mukund S; Amgen Research, South San Francisco, California., Allen JR; Amgen Research, Thousand Oaks, California., DeVoss J; Amgen Research, South San Francisco, California., Coxon A; Amgen Research, Thousand Oaks, California., Rodon J; MD Anderson, Houston, Texas., Ghiringhelli F; Centre Georges François Leclerc, Dijon, France., Penel N; Centre Oscar Lambret, Lille, France., Prenen H; Universitair Ziekenhuis Antwerpen, Edegem, Belgium., Glad S; Amgen Research, Copenhagen, Denmark., Chuang CH; Amgen Research, South San Francisco, California., Keyvanjah K; Amgen Research, Thousand Oaks, California., Townsley DM; Amgen Research, Thousand Oaks, California., Butler JR; Amgen Research, Thousand Oaks, California., Bourbeau MP; Amgen Research, Thousand Oaks, California., Caenepeel S; Amgen Research, Thousand Oaks, California., Hughes PE; Amgen Research, Thousand Oaks, California.
Source: Cancer discovery [Cancer Discov] 2025 Jan 13; Vol. 15 (1), pp. 139-161.
Publication Type: Journal Article
Journal Info: Publisher: American Association for Cancer Research Country of Publication: United States NLM ID: 101561693 Publication Model: Print Cited Medium: Internet ISSN: 2159-8290 (Electronic) Linking ISSN: 21598274 NLM ISO Abbreviation: Cancer Discov Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2159-8290
DOI:10.1158/2159-8290.CD-24-0887