Combined Inhibition of MNK Signaling and BET Proteins Reveals TGM2 as a Novel Vulnerability in Melanoma.

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Title: Combined Inhibition of MNK Signaling and BET Proteins Reveals TGM2 as a Novel Vulnerability in Melanoma.
Authors: Méant A; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada., Moussa O; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada., Lebeau B; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada; School of Biological Sciences, Nanyang Technological University, Singapore, Singapore., Gonçalves C; Lady Davis Institute, Jewish General Hospital, Montréal, Canada., Richard VR; Segal Cancer Proteomics Centre, Lady Davis Institute, Jewish General Hospital, McGill University, Montréal, Canada., Cai F; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada., Prabhu SA; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada., Langke M; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada., Guettler EM; Lady Davis Institute, Jewish General Hospital, Montréal, Canada., Su J; Lady Davis Institute, Jewish General Hospital, Montréal, Canada., Gagnon N; Lady Davis Institute, Jewish General Hospital, Montréal, Canada., Zahedi RP; Segal Cancer Proteomics Centre, Lady Davis Institute, Jewish General Hospital, McGill University, Montréal, Canada; Manitoba Centre for Proteomics and Systems Biology, University of Manitoba, Winnipeg, Canada., Borchers CH; Segal Cancer Proteomics Centre, Lady Davis Institute, Jewish General Hospital, McGill University, Montréal, Canada; Department of Oncology, McGill University, Montréal, Canada., Miller WH Jr; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada; Department of Oncology, McGill University, Montréal, Canada., Del Rincón SV; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada; Department of Oncology, McGill University, Montréal, Canada. Electronic address: soniavictoria.delrincon@mcgill.ca., Witcher M; Lady Davis Institute, Jewish General Hospital, Montréal, Canada; Division of Experimental Medicine, Department of Medicine, McGill University, Montréal, Canada; Department of Oncology, McGill University, Montréal, Canada. Electronic address: michael.witcher@mcgill.ca.
Source: The Journal of investigative dermatology [J Invest Dermatol] 2025 Apr; Vol. 145 (4), pp. 979-984.e5. Date of Electronic Publication: 2024 Oct 01.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 0426720 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1523-1747 (Electronic) Linking ISSN: 0022202X NLM ISO Abbreviation: J Invest Dermatol Subsets: MEDLINE; In Process
Database: MEDLINE Ultimate
Description
ISSN:1523-1747
DOI:10.1016/j.jid.2024.07.037