Intranasal trimethyl chitosan-coated emulsomes containing tizanidine as brain-targeted therapy in spasticity: formulation, optimization, and pharmacokinetic assessment.

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Title: Intranasal trimethyl chitosan-coated emulsomes containing tizanidine as brain-targeted therapy in spasticity: formulation, optimization, and pharmacokinetic assessment.
Authors: Elkomy MH; Department of Pharmaceutics, College of Pharmacy, Jouf University, 72341, Sakaka, Saudi Arabia., Hendawy OM; Department of Pharmacology, College of Pharmacy, Jouf University, 72341, Sakaka, Saudi Arabia. omhendawy@ju.edu.sa., Zaki RM; Department of Pharmaceutics, College of Pharmacy, Prince Sattam Bin Abdulaziz University, P.O. Box 173, 11942, Al-Kharj, Saudi Arabia.; Department of Pharmaceutics and Industrial Pharmacy, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, 62511, Egypt., Tulbah AS; Department of Pharmaceutical Sciences, College of Pharmacy, Umm Al Qura University, 21955, Makkah, Saudi Arabia., Aldosari BN; Department of Pharmaceutics, College of Pharmacy, King Saud University, P.O. Box 2457, 11451, Riyadh, Saudi Arabia., Ali AA; Department of Pharmaceutics and Industrial Pharmacy, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, 62511, Egypt., Eid HM; Department of Pharmaceutics and Industrial Pharmacy, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, 62511, Egypt. hussien.eid@pharm.bsu.edu.eg.
Source: Drug delivery and translational research [Drug Deliv Transl Res] 2025 Jul; Vol. 15 (7), pp. 2565-2580. Date of Electronic Publication: 2024 Dec 12.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Springer Country of Publication: United States NLM ID: 101540061 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2190-3948 (Electronic) Linking ISSN: 2190393X NLM ISO Abbreviation: Drug Deliv Transl Res Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:2190-3948
DOI:10.1007/s13346-024-01753-0