Synthesis and evaluation of 5, 6-dihydro-8H-isoquinolino[1, 2-b]quinazolin-8-one derivatives as novel non-lipogenic ABCA1 up-regulators with inhibitory effects on macrophage-derived foam cell formation.

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Title: Synthesis and evaluation of 5, 6-dihydro-8H-isoquinolino[1, 2-b]quinazolin-8-one derivatives as novel non-lipogenic ABCA1 up-regulators with inhibitory effects on macrophage-derived foam cell formation.
Authors: Yang C; School of Bioengineering, Zunyi Medical University, Zhuhai, China., Chen L; School of Bioengineering, Zunyi Medical University, Zhuhai, China., Jiang Y; School of Bioengineering, Zunyi Medical University, Zhuhai, China., Sun D; School of Bioengineering, Zunyi Medical University, Zhuhai, China., Hu Y; School of Bioengineering, Zunyi Medical University, Zhuhai, China.
Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2025 Dec; Vol. 40 (1), pp. 2470310. Date of Electronic Publication: 2025 Feb 26.
Publication Type: Journal Article
Journal Info: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1475-6374 (Electronic) Linking ISSN: 14756366 NLM ISO Abbreviation: J Enzyme Inhib Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1475-6374
DOI:10.1080/14756366.2025.2470310