Efficacy of MEDI0618, a pH-dependent monoclonal antibody targeting PAR2, in preclinical models of migraine.

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Title: Efficacy of MEDI0618, a pH-dependent monoclonal antibody targeting PAR2, in preclinical models of migraine.
Authors: Kopruszinski CM; Department of Pharmacology, College of Medicine, University of Arizona, Tucson, AZ 85724, USA., Linley JE; Neuroscience, BioPharmaceutical R&D, AstraZeneca, Cambridge, CB2 0AA, UK., Thornton P; Neuroscience, BioPharmaceutical R&D, AstraZeneca, Cambridge, CB2 0AA, UK., Walker AS; Neuroscience, BioPharmaceutical R&D, AstraZeneca, Cambridge, CB2 0AA, UK., Newton P; Discovery Sciences, AstraZeneca, Cambridge, CB2 0AA, UK., Podichetty S; Discovery Sciences, AstraZeneca, Cambridge, CB2 0AA, UK., Ruparel RH; Department of Pharmacology, College of Medicine, University of Arizona, Tucson, AZ 85724, USA., Moreira de Souza LH; Department of Pharmacology, College of Medicine, University of Arizona, Tucson, AZ 85724, USA., Navratilova E; Department of Pharmacology, College of Medicine, University of Arizona, Tucson, AZ 85724, USA.; Department of Neurology, Mayo Clinic, Phoenix, AZ 85054, USA., Meno-Tetang G; Neuroscience, BioPharmaceutical R&D, AstraZeneca, Cambridge, CB2 0AA, UK., Gurrell I; Neuroscience, BioPharmaceutical R&D, AstraZeneca, Cambridge, CB2 0AA, UK., Dodick DW; Department of Neurology, Mayo Clinic, Phoenix, AZ 85054, USA.; Atria Academy of Science and Medicine, New York, NY 10022, USA., Dobson C; Discovery Sciences, AstraZeneca, Cambridge, CB2 0AA, UK., Chessell T; Neuroscience, BioPharmaceutical R&D, AstraZeneca, Cambridge, CB2 0AA, UK., Porreca F; Department of Pharmacology, College of Medicine, University of Arizona, Tucson, AZ 85724, USA.; Department of Neurology, Mayo Clinic, Phoenix, AZ 85054, USA., Chessell I; Neuroscience, BioPharmaceutical R&D, AstraZeneca, Cambridge, CB2 0AA, UK.
Source: Brain : a journal of neurology [Brain] 2025 Apr 03; Vol. 148 (4), pp. 1345-1359.
Publication Type: Journal Article
Journal Info: Publisher: Oxford University Press Country of Publication: England NLM ID: 0372537 Publication Model: Print Cited Medium: Internet ISSN: 1460-2156 (Electronic) Linking ISSN: 00068950 NLM ISO Abbreviation: Brain Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1460-2156
DOI:10.1093/brain/awae344