Development of Next-Generation Antimalarial Acridones with Radical Cure Potential.

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Title: Development of Next-Generation Antimalarial Acridones with Radical Cure Potential.
Authors: Dodean RA; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States.; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States., Li Y; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States., Zhang X; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States., Caridha D; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Madejczyk MS; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Jin X; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Dennis WE; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Chetree R; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Kudyba K; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., McEnearney S; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Lee PJ; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Blount C; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., DeLuca J; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Vuong C; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Pannone K; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Dinh HT; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Mdaki K; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Leed S; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Martin ML; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Pybus BS; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Pou S; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States., Winter RW; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States., Liebman KM; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States., Williams R; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States., Kumar A; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States., Chim-Ong A; Department of Internal Medicine, Morsani College of Medicine, University of South Florida, Tampa, Florida 33612, United States., Cui L; Department of Internal Medicine, Morsani College of Medicine, University of South Florida, Tampa, Florida 33612, United States., Orena S; Infectious Diseases Research Collaboration, Kampala, Uganda., Assimwe J; Infectious Diseases Research Collaboration, Kampala, Uganda., Tibagambirwa I; Infectious Diseases Research Collaboration, Kampala, Uganda., Byaruhanga O; Infectious Diseases Research Collaboration, Kampala, Uganda., Angutoko P; Infectious Diseases Research Collaboration, Kampala, Uganda., Legac J; Department of Medicine, University of California San Francisco, San Francisco, California 94143, United States., Kreutzfeld O; Department of Medicine, University of California San Francisco, San Francisco, California 94143, United States., Rosenthal PJ; Department of Medicine, University of California San Francisco, San Francisco, California 94143, United States., Cooper RA; Department of Natural Sciences and Mathematics, Dominican University of California, San Rafael, California 94901, United States., Nilsen A; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States.; Chemical Physiology and Biochemistry, Oregon Health & Science University, Portland, Oregon 97239, United States., Riscoe MK; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States.; Molecular Microbiology and Immunology, Oregon Health & Science University, Portland, Oregon 97239, United States., Roth A; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Kancharla P; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States., Kelly JX; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States.; Department of Veterans Affairs Medical Center, Portland, Oregon 97239, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2025 Apr 24; Vol. 68 (8), pp. 8817-8840. Date of Electronic Publication: 2025 Apr 03.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.5c00419