Evidence for effective suppression of INa and IK(DR) by AS2034178 (bis{2-[(4-{(4'-(2-hydroxyethoxy)-2'-methyl[1,1'-biphenyl]-3-yl)methoxy}phenyl]methyl]-3,5-dioxo-1,2,4-oxadiazolidin-4-ide} tetrahydrate), an agonist of free fatty acid receptor.

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Title: Evidence for effective suppression of INa and IK(DR) by AS2034178 (bis{2-[(4-{(4'-(2-hydroxyethoxy)-2'-methyl[1,1'-biphenyl]-3-yl)methoxy}phenyl]methyl]-3,5-dioxo-1,2,4-oxadiazolidin-4-ide} tetrahydrate), an agonist of free fatty acid receptor.
Authors: Chou CJ; Department of Emergency Medicine, An Nan Hospital, China Medical University, Tainan 70965, Taiwan. Electronic address: 023924@tool.caaumed.org.tw., Cheung CW; Department of Anaesthesia, The University of Hong Kong, Hong Kong, China; Department of Anaesthesia, Hong Kong Sanatorium and Hospital, Hong Kong, China. Electronic address: cheucw@hku.hk., Lee CC; Department of Anaesthesia, An Nan Hospital, China Medical University, Tainan 70965, Taiwan. Electronic address: 073077@tool.caaumed.org.tw., Wu SN; Department of Physiology Cheng Kung University Medical College, Tainan 701, Taiwan; School of Medicine, National Sun Yat-Sen University College of Medicine, Kaohsiung 804, Taiwan; Department of Medical Education and Research, An Nan Hospital, China Medical University, Tainan, Taiwan. Electronic address: 071320@tool.caaumed.org.tw., Liutkeviciene R; Neuroscience Institute, Lithuanian University of Health Sciences, Kaunas, Lietuva, Lithuania. Electronic address: rasa.liukeviciene@lsmuni.lt., Rovite V; Latvian Biomedical Research and Study center, Ratsupites str 1-k1, Riga LV-1067, Latvia. Electronic address: vita.rovite@biomed.lu.lv., So EC; Department of Anaesthesia, The University of Hong Kong, Hong Kong, China; Department of Anaesthesia, An Nan Hospital, China Medical University, Tainan 70965, Taiwan. Electronic address: 011320@tool.caaumed.org.tw.
Source: Neuroscience letters [Neurosci Lett] 2025 Apr 23; Vol. 855, pp. 138222. Date of Electronic Publication: 2025 Apr 01.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Scientific Publishers Ireland Country of Publication: Ireland NLM ID: 7600130 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-7972 (Electronic) Linking ISSN: 03043940 NLM ISO Abbreviation: Neurosci Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1872-7972
DOI:10.1016/j.neulet.2025.138222