α6GABAA receptor positive allosteric modulators targeting trigeminal ganglia for preventing and aborting chronic periorbital allodynia and cephalic pain in both sexes: A mechanistic and comparative preclinical study.

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Title: α6GABAA receptor positive allosteric modulators targeting trigeminal ganglia for preventing and aborting chronic periorbital allodynia and cephalic pain in both sexes: A mechanistic and comparative preclinical study.
Authors: Chang XC; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan., Yeh CJ; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan., Pan YT; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan., Chen YP; Master of Science Degree Program in Innovation for Smart Medicine, Chang Gung University, Taoyuan City 333, Taiwan; Division of Rheumatology, Allergy and Immunology, Chang Gung Memorial Hospital at Linkou, Taoyuan City 333, Taiwan., Sharmin D; Department of Chemistry and Biochemistry, Milwaukee Institute for Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, WI 53211, USA., Cook J; Department of Chemistry and Biochemistry, Milwaukee Institute for Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, WI 53211, USA., Pei YC; Master of Science Degree Program in Innovation for Smart Medicine, Chang Gung University, Taoyuan City 333, Taiwan; Department of Physical Medicine and Rehabilitation, Chang Gung Memorial Hospital at Linkou, Taoyuan City 333, Taiwan., Chiou LC; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan; Graduate Institute of Brain and Mind Sciences, College of Medicine, National Taiwan University, Taipei 10051, Taiwan; Graduate Institute of Acupuncture Science, China Medical University, Taichung 40402, Taiwan. Electronic address: lcchiou@ntu.edu.tw.
Source: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie [Biomed Pharmacother] 2025 Aug; Vol. 189, pp. 118344. Date of Electronic Publication: 2025 Jul 12.
Publication Type: Journal Article; Comparative Study
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 8213295 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1950-6007 (Electronic) Linking ISSN: 07533322 NLM ISO Abbreviation: Biomed Pharmacother Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1950-6007
DOI:10.1016/j.biopha.2025.118344