α6GABAA receptor positive allosteric modulators targeting trigeminal ganglia for preventing and aborting chronic periorbital allodynia and cephalic pain in both sexes: A mechanistic and comparative preclinical study.

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Title: α6GABAA receptor positive allosteric modulators targeting trigeminal ganglia for preventing and aborting chronic periorbital allodynia and cephalic pain in both sexes: A mechanistic and comparative preclinical study.
Authors: Chang XC; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan., Yeh CJ; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan., Pan YT; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan., Chen YP; Master of Science Degree Program in Innovation for Smart Medicine, Chang Gung University, Taoyuan City 333, Taiwan; Division of Rheumatology, Allergy and Immunology, Chang Gung Memorial Hospital at Linkou, Taoyuan City 333, Taiwan., Sharmin D; Department of Chemistry and Biochemistry, Milwaukee Institute for Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, WI 53211, USA., Cook J; Department of Chemistry and Biochemistry, Milwaukee Institute for Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, WI 53211, USA., Pei YC; Master of Science Degree Program in Innovation for Smart Medicine, Chang Gung University, Taoyuan City 333, Taiwan; Department of Physical Medicine and Rehabilitation, Chang Gung Memorial Hospital at Linkou, Taoyuan City 333, Taiwan., Chiou LC; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan; Graduate Institute of Brain and Mind Sciences, College of Medicine, National Taiwan University, Taipei 10051, Taiwan; Graduate Institute of Acupuncture Science, China Medical University, Taichung 40402, Taiwan. Electronic address: lcchiou@ntu.edu.tw.
Source: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie [Biomed Pharmacother] 2025 Aug; Vol. 189, pp. 118344. Date of Electronic Publication: 2025 Jul 12.
Publication Type: Journal Article; Comparative Study
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 8213295 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1950-6007 (Electronic) Linking ISSN: 07533322 NLM ISO Abbreviation: Biomed Pharmacother Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: α6GABA<subscript>A</subscript> receptor positive allosteric modulators targeting trigeminal ganglia for preventing and aborting chronic periorbital allodynia and cephalic pain in both sexes: A mechanistic and comparative preclinical study.
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  Data: <searchLink fieldCode="AU" term="%22Chang+XC%22">Chang XC</searchLink>; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan.<br /><searchLink fieldCode="AU" term="%22Yeh+CJ%22">Yeh CJ</searchLink>; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan.<br /><searchLink fieldCode="AU" term="%22Pan+YT%22">Pan YT</searchLink>; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan.<br /><searchLink fieldCode="AU" term="%22Chen+YP%22">Chen YP</searchLink>; Master of Science Degree Program in Innovation for Smart Medicine, Chang Gung University, Taoyuan City 333, Taiwan; Division of Rheumatology, Allergy and Immunology, Chang Gung Memorial Hospital at Linkou, Taoyuan City 333, Taiwan.<br /><searchLink fieldCode="AU" term="%22Sharmin+D%22">Sharmin D</searchLink>; Department of Chemistry and Biochemistry, Milwaukee Institute for Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, WI 53211, USA.<br /><searchLink fieldCode="AU" term="%22Cook+J%22">Cook J</searchLink>; Department of Chemistry and Biochemistry, Milwaukee Institute for Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, WI 53211, USA.<br /><searchLink fieldCode="AU" term="%22Pei+YC%22">Pei YC</searchLink>; Master of Science Degree Program in Innovation for Smart Medicine, Chang Gung University, Taoyuan City 333, Taiwan; Department of Physical Medicine and Rehabilitation, Chang Gung Memorial Hospital at Linkou, Taoyuan City 333, Taiwan.<br /><searchLink fieldCode="AU" term="%22Chiou+LC%22">Chiou LC</searchLink>; Graduate Institute of Pharmacology, College of Medicine, National Taiwan University, Taipei 10051, Taiwan; Graduate Institute of Brain and Mind Sciences, College of Medicine, National Taiwan University, Taipei 10051, Taiwan; Graduate Institute of Acupuncture Science, China Medical University, Taichung 40402, Taiwan. Electronic address: lcchiou@ntu.edu.tw.
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  Data: <searchLink fieldCode="JN" term="%228213295%22">Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie</searchLink> [Biomed Pharmacother] 2025 Aug; Vol. 189, pp. 118344. <i>Date of Electronic Publication: </i>2025 Jul 12.
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  Data: Journal Article; Comparative Study
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Editions+Scientifiques+Elsevier%22">Editions Scientifiques Elsevier </searchLink><i>Country of Publication: </i>France <i>NLM ID: </i>8213295 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1950-6007 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2207533322%22">07533322 </searchLink><i>NLM ISO Abbreviation: </i>Biomed Pharmacother <i>Subsets: </i>MEDLINE
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        Value: 10.1016/j.biopha.2025.118344
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        Text: English
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      – TitleFull: α6GABAA receptor positive allosteric modulators targeting trigeminal ganglia for preventing and aborting chronic periorbital allodynia and cephalic pain in both sexes: A mechanistic and comparative preclinical study.
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              Text: 2025 Aug
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