Design, Synthesis, Biological Evaluation, and Computational Studies of Novel 1,4-Diketopiperazines as GABA Agonist.

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Title: Design, Synthesis, Biological Evaluation, and Computational Studies of Novel 1,4-Diketopiperazines as GABA Agonist.
Authors: Anwar MAE; Pharmaceutical Chemistry Department, Collage of Pharmaceutical Science and Drug Manufacturing, Misr University for Science and Technology, Giza, Egypt., Mohammed ER; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt., El Moghazy SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt., Abo El Nasr NME; Department of Pharmacology, National Research Centre, Medical Research and Clinical Studies Institute, Giza, Egypt., Elbaset MA; Department of Pharmacology, National Research Centre, Medical Research and Clinical Studies Institute, Giza, Egypt.; Neurology Department, Indiana University School of Medicine, Indiana, Indianapolis, USA., Korany RMS; Department of Pathology, Faculty of Veterinary Medicine, Cairo University, Giza, Egypt., Ahmed-Farid O; Department of Physiology, National Organization for Drug Control and Research, Giza, Egypt., Ibrahim IM; Biophysics Department, Faculty of Science, Cairo University, Giza, Egypt., Abd-Allah WH; Pharmaceutical Chemistry Department, Collage of Pharmaceutical Science and Drug Manufacturing, Misr University for Science and Technology, Giza, Egypt.
Source: Drug development research [Drug Dev Res] 2025 Aug; Vol. 86 (5), pp. e70136.
Publication Type: Journal Article
Journal Info: Publisher: Wiley-Liss Country of Publication: United States NLM ID: 8204468 Publication Model: Print Cited Medium: Internet ISSN: 1098-2299 (Electronic) Linking ISSN: 02724391 NLM ISO Abbreviation: Drug Dev Res Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1098-2299
DOI:10.1002/ddr.70136