Design, Synthesis, Biological Evaluation, and Computational Studies of Novel 1,4-Diketopiperazines as GABA Agonist.
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| Title: | Design, Synthesis, Biological Evaluation, and Computational Studies of Novel 1,4-Diketopiperazines as GABA Agonist. |
|---|---|
| Authors: | Anwar MAE; Pharmaceutical Chemistry Department, Collage of Pharmaceutical Science and Drug Manufacturing, Misr University for Science and Technology, Giza, Egypt., Mohammed ER; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt., El Moghazy SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt., Abo El Nasr NME; Department of Pharmacology, National Research Centre, Medical Research and Clinical Studies Institute, Giza, Egypt., Elbaset MA; Department of Pharmacology, National Research Centre, Medical Research and Clinical Studies Institute, Giza, Egypt.; Neurology Department, Indiana University School of Medicine, Indiana, Indianapolis, USA., Korany RMS; Department of Pathology, Faculty of Veterinary Medicine, Cairo University, Giza, Egypt., Ahmed-Farid O; Department of Physiology, National Organization for Drug Control and Research, Giza, Egypt., Ibrahim IM; Biophysics Department, Faculty of Science, Cairo University, Giza, Egypt., Abd-Allah WH; Pharmaceutical Chemistry Department, Collage of Pharmaceutical Science and Drug Manufacturing, Misr University for Science and Technology, Giza, Egypt. |
| Source: | Drug development research [Drug Dev Res] 2025 Aug; Vol. 86 (5), pp. e70136. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Wiley-Liss Country of Publication: United States NLM ID: 8204468 Publication Model: Print Cited Medium: Internet ISSN: 1098-2299 (Electronic) Linking ISSN: 02724391 NLM ISO Abbreviation: Drug Dev Res Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 40785696 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Design, Synthesis, Biological Evaluation, and Computational Studies of Novel 1,4-Diketopiperazines as GABA Agonist. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Anwar+MAE%22">Anwar MAE</searchLink>; Pharmaceutical Chemistry Department, Collage of Pharmaceutical Science and Drug Manufacturing, Misr University for Science and Technology, Giza, Egypt.<br /><searchLink fieldCode="AU" term="%22Mohammed+ER%22">Mohammed ER</searchLink>; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt.<br /><searchLink fieldCode="AU" term="%22El+Moghazy+SM%22">El Moghazy SM</searchLink>; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt.<br /><searchLink fieldCode="AU" term="%22Abo+El+Nasr+NME%22">Abo El Nasr NME</searchLink>; Department of Pharmacology, National Research Centre, Medical Research and Clinical Studies Institute, Giza, Egypt.<br /><searchLink fieldCode="AU" term="%22Elbaset+MA%22">Elbaset MA</searchLink>; Department of Pharmacology, National Research Centre, Medical Research and Clinical Studies Institute, Giza, Egypt.; Neurology Department, Indiana University School of Medicine, Indiana, Indianapolis, USA.<br /><searchLink fieldCode="AU" term="%22Korany+RMS%22">Korany RMS</searchLink>; Department of Pathology, Faculty of Veterinary Medicine, Cairo University, Giza, Egypt.<br /><searchLink fieldCode="AU" term="%22Ahmed-Farid+O%22">Ahmed-Farid O</searchLink>; Department of Physiology, National Organization for Drug Control and Research, Giza, Egypt.<br /><searchLink fieldCode="AU" term="%22Ibrahim+IM%22">Ibrahim IM</searchLink>; Biophysics Department, Faculty of Science, Cairo University, Giza, Egypt.<br /><searchLink fieldCode="AU" term="%22Abd-Allah+WH%22">Abd-Allah WH</searchLink>; Pharmaceutical Chemistry Department, Collage of Pharmaceutical Science and Drug Manufacturing, Misr University for Science and Technology, Giza, Egypt. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%228204468%22">Drug development research</searchLink> [Drug Dev Res] 2025 Aug; Vol. 86 (5), pp. e70136. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley-Liss%22">Wiley-Liss </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>8204468 <i>Publication Model: </i>Print <i>Cited Medium: </i>Internet <i>ISSN: </i>1098-2299 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2202724391%22">02724391 </searchLink><i>NLM ISO Abbreviation: </i>Drug Dev Res <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=40785696 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1002/ddr.70136 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: e70136 Titles: – TitleFull: Design, Synthesis, Biological Evaluation, and Computational Studies of Novel 1,4-Diketopiperazines as GABA Agonist. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Anwar MAE – PersonEntity: Name: NameFull: Mohammed ER – PersonEntity: Name: NameFull: El Moghazy SM – PersonEntity: Name: NameFull: Abo El Nasr NME – PersonEntity: Name: NameFull: Elbaset MA – PersonEntity: Name: NameFull: Korany RMS – PersonEntity: Name: NameFull: Ahmed-Farid O – PersonEntity: Name: NameFull: Ibrahim IM – PersonEntity: Name: NameFull: Abd-Allah WH IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 08 Text: 2025 Aug Type: published Y: 2025 Identifiers: – Type: issn-electronic Value: 1098-2299 Numbering: – Type: volume Value: 86 – Type: issue Value: 5 Titles: – TitleFull: Drug development research Type: main |
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