MK-8527 is a novel inhibitor of HIV-1 reverse transcriptase translocation with potential for extended-duration dosing.
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| Title: | MK-8527 is a novel inhibitor of HIV-1 reverse transcriptase translocation with potential for extended-duration dosing. |
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| Authors: | Raheem IT; Merck & Co., Inc., Rahway, New Jersey, United States of America., Girijavallabhan V; Merck & Co., Inc., Rahway, New Jersey, United States of America., Fillgrove KL; Merck & Co., Inc., Rahway, New Jersey, United States of America., Goh SL; Merck & Co., Inc., Rahway, New Jersey, United States of America., Bahnck-Teets C; Merck & Co., Inc., Rahway, New Jersey, United States of America., Huang Q; Merck & Co., Inc., Rahway, New Jersey, United States of America., Li F; Merck & Co., Inc., Rahway, New Jersey, United States of America., Wan BL; Merck & Co., Inc., Rahway, New Jersey, United States of America., O'Donnell GT; Merck & Co., Inc., Rahway, New Jersey, United States of America., Patteson JB; Merck & Co., Inc., Rahway, New Jersey, United States of America., Cilento ME; Merck & Co., Inc., Rahway, New Jersey, United States of America., Bennet A; Merck & Co., Inc., Rahway, New Jersey, United States of America., Hayes RP; Merck & Co., Inc., Rahway, New Jersey, United States of America., Tummala S; Merck & Co., Inc., Rahway, New Jersey, United States of America., McHale C; Merck & Co., Inc., Rahway, New Jersey, United States of America., Wiltsie J; Merck & Co., Inc., Rahway, New Jersey, United States of America., Ellis J; Merck & Co., Inc., Rahway, New Jersey, United States of America., Asante-Appiah E; Merck & Co., Inc., Rahway, New Jersey, United States of America., Hazuda DJ; Merck & Co., Inc., Rahway, New Jersey, United States of America., Hale J; Merck & Co., Inc., Rahway, New Jersey, United States of America., Grobler JA; Merck & Co., Inc., Rahway, New Jersey, United States of America., Xu M; Merck & Co., Inc., Rahway, New Jersey, United States of America., Diamond TL; Merck & Co., Inc., Rahway, New Jersey, United States of America., Lai MT; Merck & Co., Inc., Rahway, New Jersey, United States of America. |
| Source: | PLoS biology [PLoS Biol] 2025 Aug 26; Vol. 23 (8), pp. e3003308. Date of Electronic Publication: 2025 Aug 26 (Print Publication: 2025). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Public Library of Science Country of Publication: United States NLM ID: 101183755 Publication Model: eCollection Cited Medium: Internet ISSN: 1545-7885 (Electronic) Linking ISSN: 15449173 NLM ISO Abbreviation: PLoS Biol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| ISSN: | 1545-7885 |
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| DOI: | 10.1371/journal.pbio.3003308 |