Molecular docking-based design of novel tricyclic tetrahydropyridothienopyrimidinone derivatives as AChE/MAO-B dual inhibitors.

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Title: Molecular docking-based design of novel tricyclic tetrahydropyridothienopyrimidinone derivatives as AChE/MAO-B dual inhibitors.
Authors: Zhang J; Center of Safety Evaluation and Research, Hangzhou Medical College, Hangzhou, 310013, Zhejiang, China.; School of Biological Science and Technology, University of Jinan, Jinan, 250022, China., Li Y; School of Biological Science and Technology, University of Jinan, Jinan, 250022, China.; Advanced Medical Research Institute, Cheeloo College of Medicine, Shandong University, Jinan, 250012, Shandong, China., Shao JD; Advanced Medical Research Institute, Cheeloo College of Medicine, Shandong University, Jinan, 250012, Shandong, China., Wei G; School of Biological Science and Technology, University of Jinan, Jinan, 250022, China., Zhang NY; School of Biological Science and Technology, University of Jinan, Jinan, 250022, China., Zhu KK; Advanced Medical Research Institute, Cheeloo College of Medicine, Shandong University, Jinan, 250012, Shandong, China., Wang KM; School of Biological Science and Technology, University of Jinan, Jinan, 250022, China. bio_wangkm@ujn.edu.cn., Jiang CS; School of Biological Science and Technology, University of Jinan, Jinan, 250022, China. bio_jiangcs@ujn.edu.cn., Wang JH; Center of Safety Evaluation and Research, Hangzhou Medical College, Hangzhou, 310013, Zhejiang, China. jhongwang89@163.com.
Source: Molecular diversity [Mol Divers] 2026 Jun; Vol. 30 (3), pp. 4121-4136. Date of Electronic Publication: 2025 Sep 20.
Publication Type: Journal Article
Journal Info: Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1573-501X
DOI:10.1007/s11030-025-11354-9