Optimization of Prodiginines as Single-Dose Curative Antimalarials.

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Bibliographic Details
Title: Optimization of Prodiginines as Single-Dose Curative Antimalarials.
Authors: Kumar A; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States., Li Y; Department of Veterans Affairs Medical Center, Portland VA Medical Center as the Institution, Portland, Oregon 97239, United States., Zhang X; Department of Veterans Affairs Medical Center, Portland VA Medical Center as the Institution, Portland, Oregon 97239, United States., Gaddam M; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States., Caridha D; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Madejczyk MS; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Jin X; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Dennis WE; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Chetree R; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Blount C; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., DeLuca J; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Vuong C; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Kudyba K; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States.; Integrated Pathogen Therapeutics Department, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Roncal N; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States.; Integrated Pathogen Therapeutics Department, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Ashraf K; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States.; Integrated Pathogen Therapeutics Department, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Lee PJ; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Pannone K; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Leed S; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States.; Integrated Pathogen Therapeutics Department, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Dinh HT; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Mdaki K; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Navarrete K; Department of Natural Sciences and Mathematics, Dominican University of California, San Rafael, California 94901, United States., Charlton J; Department of Natural Sciences and Mathematics, Dominican University of California, San Rafael, California 94901, United States., Binauhan AJ; Department of Natural Sciences and Mathematics, Dominican University of California, San Rafael, California 94901, United States., Qahash T; Department of Biological Sciences, Eck Institute for Global Health, University of Notre Dame, Notre Dame, Indiana 46556, United States., Kibe KM; Department of Biological Sciences, Eck Institute for Global Health, University of Notre Dame, Notre Dame, Indiana 46556, United States., Shoue DA; Department of Biological Sciences, Eck Institute for Global Health, University of Notre Dame, Notre Dame, Indiana 46556, United States., Checkley L; Department of Biological Sciences, Eck Institute for Global Health, University of Notre Dame, Notre Dame, Indiana 46556, United States., Ferdig MT; Department of Biological Sciences, Eck Institute for Global Health, University of Notre Dame, Notre Dame, Indiana 46556, United States., Chim-Ong A; Department of Internal Medicine, Morsani College of Medicine, University of South Florida, Tampa, Florida 33612, United States., Cui L; Department of Internal Medicine, Morsani College of Medicine, University of South Florida, Tampa, Florida 33612, United States., Orena S; Infectious Diseases Research Collaboration, Kampala, Uganda., Byaruhanga O; Infectious Diseases Research Collaboration, Kampala, Uganda., Assimwe J; Infectious Diseases Research Collaboration, Kampala, Uganda., Tibagambirwa I; Infectious Diseases Research Collaboration, Kampala, Uganda., Chithanna S; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States., Dodean RA; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States.; Department of Veterans Affairs Medical Center, Portland VA Medical Center as the Institution, Portland, Oregon 97239, United States., Legac J; Department of Medicine, University of California San Francisco, San Francisco, California 94143, United States., Kreutzfeld O; Department of Medicine, University of California San Francisco, San Francisco, California 94143, United States., Rosenthal PJ; Department of Medicine, University of California San Francisco, San Francisco, California 94143, United States., Cooper RA; Department of Natural Sciences and Mathematics, Dominican University of California, San Rafael, California 94901, United States., Reynolds KA; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States., Roth A; Experimental Therapeutics Branch, CIDR, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States.; Integrated Pathogen Therapeutics Department, Walter Reed Army Institute of Research, Silver Spring, Maryland 20910, United States., Kelly JX; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States.; Department of Veterans Affairs Medical Center, Portland VA Medical Center as the Institution, Portland, Oregon 97239, United States., Kancharla P; Department of Chemistry, Portland State University, Portland, Oregon 97201, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2025 Nov 27; Vol. 68 (22), pp. 24469-24501. Date of Electronic Publication: 2025 Nov 18.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.5c02523