Mirtazapine is a functional antagonist at cardiac human H1-histamine receptors.

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Title: Mirtazapine is a functional antagonist at cardiac human H1-histamine receptors.
Authors: Pham TH; Institute for Pharmacology and Toxicology, Medical Faculty, Martin-Luther-University Halle-Wittenberg, Magdeburger Straße 4, 06097, Halle (Saale), Germany., Schlicht JMA; Institute for Pharmacology and Toxicology, Medical Faculty, Martin-Luther-University Halle-Wittenberg, Magdeburger Straße 4, 06097, Halle (Saale), Germany., Hofmann B; Department of Cardiac Surgery, Mid-German Heart Centre, University Hospital Halle, Ernst-Grube-Straße 40, 06097, Halle (Saale), Germany., Kirchhefer U; Institute for Pharmacology and Toxicology, University Hospital Münster, University Münster, Domagkstraße 12, 48149, Münster, Germany., Neumann J; Institute for Pharmacology and Toxicology, Medical Faculty, Martin-Luther-University Halle-Wittenberg, Magdeburger Straße 4, 06097, Halle (Saale), Germany. joachim.neumann@medizin.uni-halle.de., Gergs U; Institute for Pharmacology and Toxicology, Medical Faculty, Martin-Luther-University Halle-Wittenberg, Magdeburger Straße 4, 06097, Halle (Saale), Germany.
Source: Naunyn-Schmiedeberg's archives of pharmacology [Naunyn Schmiedebergs Arch Pharmacol] 2026 Mar; Vol. 399 (6), pp. 8061-8074. Date of Electronic Publication: 2025 Dec 20.
Publication Type: Journal Article
Journal Info: Publisher: Springer Verlag Country of Publication: Germany NLM ID: 0326264 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1432-1912 (Electronic) Linking ISSN: 00281298 NLM ISO Abbreviation: Naunyn Schmiedebergs Arch Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1432-1912
DOI:10.1007/s00210-025-04908-z