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BET Isoform Selectivity through Diverse Linkers for Bivalent Inhibitors: GSK785, a BRD2/4-Selective Bivalent BET Inhibitor.

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Bibliographic Details
Title:	BET Isoform Selectivity through Diverse Linkers for Bivalent Inhibitors: GSK785, a BRD2/4-Selective Bivalent BET Inhibitor.
Authors:	Rianjongdee F; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Atkinson SJ; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Bamborough P; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Barnett HA; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Friston K; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Grandi P; Cellzome, GlaxoSmithKline, Meyerhofstr. 1, Heidelberg 69117, Germany., Neipp CE; GSK, South Collegeville Road, Collegeville, Pennsylvania 19426-0989, United States., Petretich M; Cellzome, GlaxoSmithKline, Meyerhofstr. 1, Heidelberg 69117, Germany., Phillipou A; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Preston AGS; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Prinjha RK; GSK, Stevenage, Hertfordshire SG1 2NY, U.K., Tomkinson NCO; Department for Pure and Applied Chemistry, University of Strathclyde, 295 Cathedral Street, Glasgow G1 1XL, U.K., Demont EH; GSK, Stevenage, Hertfordshire SG1 2NY, U.K.
Source:	Journal of medicinal chemistry [J Med Chem] 2026 Jan 22; Vol. 69 (2), pp. 895-917. Date of Electronic Publication: 2025 Dec 30.
Publication Type:	Journal Article
Journal Info:	Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database:	MEDLINE Ultimate

Description
ISSN:	1520-4804
DOI:	10.1021/acs.jmedchem.5c00622