Epigenetic enzyme inhibitors targeting DNA, histone, and RNA methylation: Mechanisms and therapeutic applications in cancer.

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Title: Epigenetic enzyme inhibitors targeting DNA, histone, and RNA methylation: Mechanisms and therapeutic applications in cancer.
Authors: Wang Y; College of Pharmacy and Food, Southwest Minzu University, Chengdu, Sichuan, 610225, China., Ma C; College of Pharmacy and Food, Southwest Minzu University, Chengdu, Sichuan, 610225, China., Liu X; College of Pharmacy and Food, Southwest Minzu University, Chengdu, Sichuan, 610225, China., Cheng J; College of Pharmacy and Food, Southwest Minzu University, Chengdu, Sichuan, 610225, China., Zhu D; Department of Endocrinology and Nephrology, 363 Hospital, Chengdu, 610065, China., Liu P; Institute of Chemistry, Henan Academy of Sciences, Zhengzhou, Henan, 450053, China., Qi P; Institute of Chemistry, Henan Academy of Sciences, Zhengzhou, Henan, 450053, China. Electronic address: qipeng@hnas.ac.cn., Li X; Institute of Chemistry, Henan Academy of Sciences, Zhengzhou, Henan, 450053, China. Electronic address: lixiankai@hnas.ac.cn., Gu J; College of Pharmacy and Food, Southwest Minzu University, Chengdu, Sichuan, 610225, China. Electronic address: gujiancd@163.com., Wang Q; College of Pharmacy and Food, Southwest Minzu University, Chengdu, Sichuan, 610225, China; Department of Pathology, Yong Loo Lin School of Medicine, National University of Singapore, Singapore, 117597, Singapore. Electronic address: patv127@nus.edu.sg.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2026 Mar 15; Vol. 306, pp. 118590. Date of Electronic Publication: 2026 Jan 20.
Publication Type: Journal Article; Review
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1768-3254
DOI:10.1016/j.ejmech.2026.118590