Pharmacophore-Based Identification and Molecular Characterization of Potent Neprilysin Inhibitors: Biochemical and Therapeutic Implications for Cardiovascular Diseases.

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Title: Pharmacophore-Based Identification and Molecular Characterization of Potent Neprilysin Inhibitors: Biochemical and Therapeutic Implications for Cardiovascular Diseases.
Authors: Kuo CT; Department of Cardiovascular Surgery, Ditmanson Medical Foundation Chia-Yi Christian Hospital, Chiayi, Taiwan., Wu YC; Institute of Molecular Biology, National Chung Hsing University, Taichung, Taiwan., Li JM; Institute of Precision Medicine, College of Medicine, National Sun Yat-Sen University, Kaohsiung, Taiwan.; Center of Excellence for Metabolic Associated Fatty Liver Disease, National Sun Yat-Sen University, Kaohsiung, Taiwan., Ju TC; Institute of Molecular Biology, National Chung Hsing University, Taichung, Taiwan.; International Doctoral Program in Interdisciplinary Innovative Life Science and Technology, National Chung Hsing University, Taichung, Taiwan.; Doctoral Program in Translational Medicine, National Chung Hsing University, Taichung, Taiwan., Tseng TS; Institute of Molecular Biology, National Chung Hsing University, Taichung, Taiwan.; International Doctoral Program in Interdisciplinary Innovative Life Science and Technology, National Chung Hsing University, Taichung, Taiwan.; Doctoral Program in Microbial Genomics, National Chung Hsing University and Academia Sinica, Taichung, Taiwan.
Source: Chemical biology & drug design [Chem Biol Drug Des] 2026 Feb; Vol. 107 (2), pp. e70247.
Publication Type: Journal Article
Journal Info: Publisher: Wiley-Blackwell Country of Publication: England NLM ID: 101262549 Publication Model: Print Cited Medium: Internet ISSN: 1747-0285 (Electronic) Linking ISSN: 17470277 NLM ISO Abbreviation: Chem Biol Drug Des Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1747-0285
DOI:10.1111/cbdd.70247