Pharmacokinetics of Asciminib 200 mg in the Presence of a Strong CYP3A4 Inducer, Phenytoin, in Healthy Participants.

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Title: Pharmacokinetics of Asciminib 200 mg in the Presence of a Strong CYP3A4 Inducer, Phenytoin, in Healthy Participants.
Authors: Hoch M; Novartis Biomedical Research, Basel, Switzerland. matthias.hoch@novartis.com., Taylor AJ; Novartis Pharmaceuticals Corporation, East Hanover, NJ, USA., Huth F; Novartis Biomedical Research, Basel, Switzerland., Jamalapuram S; Novartis Pharmaceuticals Corporation, East Hanover, NJ, USA., Loisios-Konstantinidis I; Novartis Biomedical Research, Basel, Switzerland., Quinlan M; Novartis Pharmaceuticals Corporation, East Hanover, NJ, USA., Kranidi A; Novartis Ireland Limited, Dublin, Ireland., Coleman D; Novartis Pharma AG, Basel, Switzerland., Espurz N; Novartis Pharma AG, Basel, Switzerland., Bellibas SE; Novartis Pharmaceuticals Corporation, East Hanover, NJ, USA., Pierre AS; Novartis Biomedical Research, Basel, Switzerland.
Source: Clinical pharmacokinetics [Clin Pharmacokinet] 2026 May; Vol. 65 (5), pp. 709-718. Date of Electronic Publication: 2026 Mar 17.
Publication Type: Journal Article; Clinical Trial, Phase I
Journal Info: Publisher: Country of Publication: Switzerland NLM ID: 7606849 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1179-1926 (Electronic) Linking ISSN: 03125963 NLM ISO Abbreviation: Clin Pharmacokinet Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1179-1926
DOI:10.1007/s40262-026-01629-1