Drugging the intrinsically disordered transactivation domain of androgen receptor.
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| Title: | Drugging the intrinsically disordered transactivation domain of androgen receptor. |
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| Authors: | Obst JK; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Banuelos CA; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Jian K; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada., Tien AH; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Shkrabak OA; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada., Wang J; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Mawji NR; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Tam T; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Vuckovic M; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada., Williams DE; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada., Rogalski JC; Proteomics and Metabolomics Core Facility, Life Sciences Institute, University of British Columbia, Vancouver, BC, Canada., Yuan X; Proteomics and Metabolomics Core Facility, Life Sciences Institute, University of British Columbia, Vancouver, BC, Canada., Strynadka NCJ; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada. natalie.strynadka@ubc.ca., Andersen RJ; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada. raymond.andersen@ubc.ca., Sadar MD; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada. msadar@bcgsc.ca. |
| Source: | Signal transduction and targeted therapy [Signal Transduct Target Ther] 2026 Apr 28; Vol. 11 (1). Date of Electronic Publication: 2026 Apr 28. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101676423 Publication Model: Electronic Cited Medium: Internet ISSN: 2059-3635 (Electronic) Linking ISSN: 20593635 NLM ISO Abbreviation: Signal Transduct Target Ther Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| ISSN: | 2059-3635 |
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| DOI: | 10.1038/s41392-026-02642-3 |