Drugging the intrinsically disordered transactivation domain of androgen receptor.

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Title: Drugging the intrinsically disordered transactivation domain of androgen receptor.
Authors: Obst JK; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Banuelos CA; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Jian K; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada., Tien AH; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Shkrabak OA; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada., Wang J; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Mawji NR; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Tam T; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada., Vuckovic M; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada., Williams DE; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada., Rogalski JC; Proteomics and Metabolomics Core Facility, Life Sciences Institute, University of British Columbia, Vancouver, BC, Canada., Yuan X; Proteomics and Metabolomics Core Facility, Life Sciences Institute, University of British Columbia, Vancouver, BC, Canada., Strynadka NCJ; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada. natalie.strynadka@ubc.ca., Andersen RJ; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada. raymond.andersen@ubc.ca., Sadar MD; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada. msadar@bcgsc.ca.
Source: Signal transduction and targeted therapy [Signal Transduct Target Ther] 2026 Apr 28; Vol. 11 (1). Date of Electronic Publication: 2026 Apr 28.
Publication Type: Journal Article
Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101676423 Publication Model: Electronic Cited Medium: Internet ISSN: 2059-3635 (Electronic) Linking ISSN: 20593635 NLM ISO Abbreviation: Signal Transduct Target Ther Subsets: MEDLINE
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  Data: <searchLink fieldCode="AU" term="%22Obst+JK%22">Obst JK</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Banuelos+CA%22">Banuelos CA</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Jian+K%22">Jian K</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Tien+AH%22">Tien AH</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Shkrabak+OA%22">Shkrabak OA</searchLink>; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Wang+J%22">Wang J</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Mawji+NR%22">Mawji NR</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Tam+T%22">Tam T</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Vuckovic+M%22">Vuckovic M</searchLink>; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Williams+DE%22">Williams DE</searchLink>; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Rogalski+JC%22">Rogalski JC</searchLink>; Proteomics and Metabolomics Core Facility, Life Sciences Institute, University of British Columbia, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Yuan+X%22">Yuan X</searchLink>; Proteomics and Metabolomics Core Facility, Life Sciences Institute, University of British Columbia, Vancouver, BC, Canada.<br /><searchLink fieldCode="AU" term="%22Strynadka+NCJ%22">Strynadka NCJ</searchLink>; Dept. of Biochemistry and Molecular Biology and the Center for Blood Research, Life Sciences Centre, University of British Columbia, Vancouver, BC, Canada. natalie.strynadka@ubc.ca.<br /><searchLink fieldCode="AU" term="%22Andersen+RJ%22">Andersen RJ</searchLink>; Chemistry and Earth, Ocean and Atmospheric Sciences, University of British Columbia, Vancouver, BC, Canada. raymond.andersen@ubc.ca.<br /><searchLink fieldCode="AU" term="%22Sadar+MD%22">Sadar MD</searchLink>; Canada's Michael Smith Genome Sciences Centre at BC Cancer, Vancouver, BC, Canada. msadar@bcgsc.ca.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Nature+Publishing+Group%22">Nature Publishing Group </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>101676423 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2059-3635 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2220593635%22">20593635 </searchLink><i>NLM ISO Abbreviation: </i>Signal Transduct Target Ther <i>Subsets: </i>MEDLINE
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              Text: 2026 Apr 28
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