Identification of a Quinolone-Based Scaffold as a Dual SARS-COV-2 PLᵖʳᵒ and Mᵖʳᵒ Inhibitor: An Integrated Molecular Modeling and In-vitro Evaluation Approach.

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Title: Identification of a Quinolone-Based Scaffold as a Dual SARS-COV-2 PLᵖʳᵒ and Mᵖʳᵒ Inhibitor: An Integrated Molecular Modeling and In-vitro Evaluation Approach.
Authors: Atatreh N; College of Pharmacy, Al Ain University, Abu Dhabi, United Arab Emirates.; AAU Health and Biomedical Research Center, Al Ain University, Abu Dhabi, United Arab Emirates., Bustanji L; College of Pharmacy, Al Ain University, Abu Dhabi, United Arab Emirates.; AAU Health and Biomedical Research Center, Al Ain University, Abu Dhabi, United Arab Emirates., Ferreira JC; Science Division, New York University, Abu Dhabi, 129188, United Arab Emirates., Rabeh WM; Science Division, New York University, Abu Dhabi, 129188, United Arab Emirates., Mahgoub RE; College of Pharmacy, Al Ain University, Abu Dhabi, United Arab Emirates.; AAU Health and Biomedical Research Center, Al Ain University, Abu Dhabi, United Arab Emirates., Ghattas MA; College of Pharmacy, Al Ain University, Abu Dhabi, United Arab Emirates.; AAU Health and Biomedical Research Center, Al Ain University, Abu Dhabi, United Arab Emirates.
Source: Drug design, development and therapy [Drug Des Devel Ther] 2026 May 04; Vol. 20, pp. 593126. Date of Electronic Publication: 2026 May 04 (Print Publication: 2026).
Publication Type: Journal Article
Journal Info: Publisher: Dove Press Limited Country of Publication: New Zealand NLM ID: 101475745 Publication Model: eCollection Cited Medium: Internet ISSN: 1177-8881 (Electronic) Linking ISSN: 11778881 NLM ISO Abbreviation: Drug Des Devel Ther Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1177-8881
DOI:10.2147/DDDT.S593126