CYP3A-Mediated Metabolism of Zastaprazan in Humans and Associated Drug-Drug Interactions.

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Title: CYP3A-Mediated Metabolism of Zastaprazan in Humans and Associated Drug-Drug Interactions.
Authors: Cao KJ; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; University of Chinese Academy of Sciences, Beijing 100049, China., Fu L; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Sun YC; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China., Meng J; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China., Huang Q; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Deng DC; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Hu HT; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Han ZH; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Guo G; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China., Zhou X; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.; School of Pharmacy, Fudan University, Shanghai 200433, China., Chen XY; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; University of Chinese Academy of Sciences, Beijing 100049, China.
Source: Pharmaceutics [Pharmaceutics] 2026 Jun 10; Vol. 18 (6). Date of Electronic Publication: 2026 Jun 10.
Publication Type: Journal Article
Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101534003 Publication Model: Electronic Cited Medium: Print ISSN: 1999-4923 (Print) Linking ISSN: 19994923 NLM ISO Abbreviation: Pharmaceutics Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1999-4923
DOI:10.3390/pharmaceutics18060718