Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.

Saved in:
Bibliographic Details
Title: Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.
Authors: Deng H; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Bernier SG; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Doyle E; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Lorusso J; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Morgan BA; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Westlin WF; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States., Evindar G; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2013 Aug 27; Vol. 4 (10), pp. 942-7. Date of Electronic Publication: 2013 Aug 27 (Print Publication: 2013).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
FullText Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 24900589
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Deng+H%22">Deng H</searchLink>; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Bernier+SG%22">Bernier SG</searchLink>; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Doyle+E%22">Doyle E</searchLink>; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Lorusso+J%22">Lorusso J</searchLink>; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Morgan+BA%22">Morgan BA</searchLink>; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Westlin+WF%22">Westlin WF</searchLink>; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Evindar+G%22">Evindar G</searchLink>; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2013 Aug 27; Vol. 4 (10), pp. 942-7. <i>Date of Electronic Publication: </i>2013 Aug 27 (<i>Print Publication: </i>2013).
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=24900589
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1021/ml400194r
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 942
    Titles:
      – TitleFull: Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Deng H
      – PersonEntity:
          Name:
            NameFull: Bernier SG
      – PersonEntity:
          Name:
            NameFull: Doyle E
      – PersonEntity:
          Name:
            NameFull: Lorusso J
      – PersonEntity:
          Name:
            NameFull: Morgan BA
      – PersonEntity:
          Name:
            NameFull: Westlin WF
      – PersonEntity:
          Name:
            NameFull: Evindar G
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 27
              M: 08
              Text: 2013 Aug 27
              Type: published
              Y: 2013
          Identifiers:
            – Type: issn-print
              Value: 1948-5875
          Numbering:
            – Type: volume
              Value: 4
            – Type: issue
              Value: 10
          Titles:
            – TitleFull: ACS medicinal chemistry letters
              Type: main
ResultId 1